SCHEMBL8565751

SCHEMBL8565751

Nc1nc(N)c2c(n1)CCC2CCOc1ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)cc1

nearest known ligand 0.77

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
DHFR P00374 6/20 0.57
MTR Q99707 1/20 0.55
GART P22102 3/20 0.52
FOLR2 P14207 1/20 0.48
FOLR1 P15328 1/20 0.48
SLC19A1 P41440 1/20 0.48
SLC46A1 Q96NT5 1/20 0.48
ATIC P31939 1/20 0.47
SHMT1 P34896 1/20 0.47
SHMT2 P34897 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8571475 0.87 DHFR (0.57) DHFRMTRGART
SCHEMBL1066004 0.85 DHFR (0.59) DHFRMTRGARTATIC
SCHEMBL8571393 0.85 ATIC (0.59) DHFRMTRATIC
SCHEMBL9043308 0.85 DHFR (0.57) DHFRGARTFOLR2FOLR1SLC19A1
SCHEMBL8603963 0.85 DHFR (0.55) DHFRMTR
SCHEMBL8570088 0.83 DHFR (0.58) DHFRMTR
SCHEMBL8567642 0.81 DHFR (0.45) DHFR
SCHEMBL9001966 0.81 DHFR (0.55) DHFRMTR
SCHEMBL8569142 0.81 DHFR (0.59) DHFRMTR
SCHEMBL9001801 0.79 DHFR (0.53) DHFRMTRGARTATIC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0530579-B1 Condensed pyrimidine derivatives antitumor agents EISAI CO LTD (JP) 1998-11-11 EP disclosed
US-5554615-A ANTITUMOR EISAI CO., LTD. (JP) 1996-09-10 US disclosed
EP-0530579-A1 Condensed pyrimidine derivatives antitumor agents Eisai Co., Ltd. (JP) 1993-03-10 EP disclosed