SCHEMBL9043308

SCHEMBL9043308

Nc1nc(N)c2c(n1)NCC2CCOc1ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)cc1

nearest known ligand 0.59

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DHFR P00374 4/20 0.57
GART P22102 4/20 0.54
FOLR2 P14207 1/20 0.50
FOLR1 P15328 1/20 0.50
SLC19A1 P41440 1/20 0.50
SLC46A1 Q96NT5 1/20 0.50
ATIC P31939 2/20 0.49
SHMT1 P34896 1/20 0.49
SHMT2 P34897 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9042931 0.86 DHFR (0.60) DHFRGARTFOLR2FOLR1SLC46A1
SCHEMBL9041817 0.85 MTHFD1 (0.59) DHFRGARTATIC
SCHEMBL8997257 0.85 GART (0.61) DHFRGARTATIC
SCHEMBL9041263 0.85 DHFR (0.50) DHFRGART
SCHEMBL9041254 0.85 DHFR (0.50) DHFRGART
SCHEMBL8565751 0.85 DHFR (0.57) DHFRGARTFOLR2FOLR1SLC19A1
SCHEMBL8997170 0.85 DHFR (0.55) DHFRGARTATIC
SCHEMBL9758306 0.85 DHFR (0.55) DHFRGARTATIC
SCHEMBL9088274 0.84 ATIC (0.51) DHFRGARTATIC
SCHEMBL9227797 0.84 DHFR (0.57) DHFRGARTFOLR2FOLR1SLC46A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0400562-B1 Pyrrolopyrimidines, their production and use as tumoricidal agents TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1996-08-21 EP disclosed