SCHEMBL8566830

SCHEMBL8566830

CCCCC1n2c(c(C(N)=O)c3ccccc32)SC1(C)C1CCNCC1

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.39
HTR2C P28335 2/20 0.39
CNR2 P34972 5/20 0.34
CNR1 P21554 4/20 0.34
REN P00797 5/20 0.33
EGFR P00533 1/20 0.32
SRC P12931 1/20 0.32
HTR4 Q13639 2/20 0.32
NPC1 O15118 2/20 0.31
PARP1 P09874 1/20 0.31
PARP2 Q9UGN5 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8574553 0.84 HTR2A (0.39) HTR2AHTR2CCNR2CNR1EGFR
SCHEMBL8520380 0.79 HTR2A (0.39) HTR2AHTR2CCNR2CNR1REN
SCHEMBL8521038 0.74 HTR2A (0.41) HTR2AHTR2CCNR2CNR1EGFR
SCHEMBL1077434 0.72 HTR2A (0.39) HTR2AHTR2CCNR2CNR1EGFR
SCHEMBL8575510 0.71 HTR2A (0.41) HTR2AHTR2CCNR2HTR4
SCHEMBL8575716 0.69 HTR2A (0.38) HTR2AHTR2CCNR2HTR4
SCHEMBL8566824 0.66 HTR4 (0.47) HTR4
SCHEMBL8574546 0.65 HTR4 (0.46) HTR4
SCHEMBL7449849 0.61 KDM4E (0.53) CNR2CNR1HTR4
SCHEMBL8521031 0.60 HTR4 (0.46) CNR2CNR1HTR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5998409-A GASTROINTESTINAL DISORDERS; CARDIOVASCULAR DISORDERS; NERVOUS SYSTEM DISORDERS SMITHKLINE BEECHAM PLC (GB) 1999-12-07 US disclosed