SCHEMBL8575716

SCHEMBL8575716

CCCCCCC1Cn2c(c(C(N)=O)c3ccccc32)OC1(C)C1CCNCC1

nearest known ligand 0.38

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.38
HTR2C P28335 2/20 0.38
HTR4 Q13639 2/20 0.36
CNR2 P34972 1/20 0.32
ICMT O60725 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1077434 0.96 HTR2A (0.39) HTR2AHTR2CHTR4CNR2
SCHEMBL8575510 0.89 HTR2A (0.41) HTR2AHTR2CHTR4CNR2
SCHEMBL8520380 0.81 HTR2A (0.39) HTR2AHTR2CHTR4CNR2
SCHEMBL8521038 0.79 HTR2A (0.41) HTR2AHTR2CHTR4CNR2
SCHEMBL8574553 0.77 HTR2A (0.39) HTR2AHTR2CHTR4CNR2
SCHEMBL8575712 0.70 HTR4 (0.47) HTR2AHTR4
SCHEMBL8566830 0.69 HTR2A (0.39) HTR2AHTR2CHTR4CNR2
SCHEMBL1077431 0.68 HTR4 (0.50) HTR2AHTR4
SCHEMBL8575502 0.67 HTR4 (0.53) HTR2AHTR4
SCHEMBL8521031 0.61 HTR4 (0.46) HTR4CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5998409-A GASTROINTESTINAL DISORDERS; CARDIOVASCULAR DISORDERS; NERVOUS SYSTEM DISORDERS SMITHKLINE BEECHAM PLC (GB) 1999-12-07 US disclosed