SCHEMBL8566993

SCHEMBL8566993

[CH2]Oc1ccc2cccc(N3CCN(C)CC3)c2c1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 13/20 0.73
HTR1D P28221 10/20 0.73
HTR1B P28222 10/20 0.73
SLC6A9 P48067 1/20 0.50
KCNH2 Q12809 1/20 0.50
MTNR1B P49286 1/20 0.50
HTR3A P46098 1/20 0.49
ADRB2 P07550 2/20 0.43
ADRB1 P08588 2/20 0.43
ADRA2A P08913 2/20 0.43
DRD2 P14416 2/20 0.43
ADRA2B P18089 2/20 0.43
ADRA2C P18825 2/20 0.43
DRD1 P21728 2/20 0.43
DRD4 P21917 2/20 0.43
SLC6A2 P23975 2/20 0.43
HRH2 P25021 2/20 0.43
ADRA1D P25100 2/20 0.43
HTR2A P28223 2/20 0.43
HTR2C P28335 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6000211 0.87 HTR1A (0.75) HTR1AHTR1DHTR1BSLC6A9KCNH2
SCHEMBL9062634 0.81 HTR1A (0.81) HTR1AHTR1DHTR1BSLC6A9KCNH2
SCHEMBL6313399 0.80 HTR1A (0.69) HTR1AHTR1DHTR1BSLC6A9KCNH2
SCHEMBL6314991 0.80 HTR1A (0.64) HTR1AHTR1DHTR1BSLC6A9KCNH2
SCHEMBL6312894 0.79 HTR1A (0.75) HTR1AHTR1DHTR1BSLC6A9KCNH2
SCHEMBL6313298 0.79 HTR1A (0.63) HTR1AHTR1DHTR1BHTR3AADRB2
SCHEMBL6307480 0.78 HTR1A (0.62) HTR1AHTR1DHTR1BSLC6A9KCNH2
SCHEMBL9058520 0.78 HTR1A (0.79) HTR1AHTR1DHTR1BSLC6A9KCNH2
SCHEMBL9058908 0.78 HTR1A (0.81) HTR1AHTR1DHTR1BSLC6A9KCNH2
SCHEMBL9054738 0.78 HTR1A (0.81) HTR1AHTR1DHTR1BSLC6A9KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5821245-A Use of naphthalene derivatives in treating lung carcinoma PFIZER INC. (US) 1998-10-13 US disclosed