SCHEMBL8567342

SCHEMBL8567342

CCOC(=O)COc1ccc(C(C#N)CCCCCOc2cc(OCc3ccccc3)c(Br)cc2CC)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 3/20 0.39
ESR1 P03372 1/20 0.38
HPGD P15428 2/20 0.38
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
TP53 P04637 1/20 0.38
MAPT P10636 1/20 0.38
HSD17B10 Q99714 1/20 0.38
CCR1 P32246 1/20 0.36
FFAR1 O14842 2/20 0.36
PPARG P37231 1/20 0.36
PPARA Q07869 1/20 0.36
NPC1 O15118 1/20 0.36
MAPK1 P28482 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
LTA4H P09960 1/20 0.36
LMNA P02545 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
ABCB1 P08183 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8561236 0.89 FFAR1 (0.40) NR1H4ESR1HPGDKDM4EALDH1A1
SCHEMBL8565242 0.87 LTB4R (0.39) NR1H4ESR1HPGDKDM4EALDH1A1
SCHEMBL8562772 0.87 NR1H4 (0.43) NR1H4ALDH1A1CCR1RAB9ALMNA
SCHEMBL8565673 0.83 MAOB (0.43) NR1H4HPGDMAPTCCR1FFAR1
SCHEMBL9226094 0.82 NR1H4 (0.35) NR1H4CCR1FFAR1LMNAABCB1
SCHEMBL8564071 0.76 SGMS2 (0.41) NR1H4CCR1FFAR1
SCHEMBL8561446 0.74 GAA (0.46) HPGDKDM4EALDH1A1TP53MAPT
SCHEMBL8562831 0.73 PTGER1 (0.46)
SCHEMBL8567408 0.73 GAA (0.45) HPGDKDM4EALDH1A1TP53MAPT
SCHEMBL6762521 0.73 NR1H4 (0.44) NR1H4LMNAPTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0544488-B1 Substituted phenyl phenol leukotriene antagonists LILLY CO ELI (US) 1998-03-11 EP disclosed
WO-1996036347-A1 USE OF LEUKOTRIENE ANTAGONISTS FOR ALZHEIMER'S DISEASE ELI LILLY AND COMPANY (US) 1996-11-21 WO disclosed
EP-0743064-A1 Leukotriene antagonists for use in the treatment or prevention of alzheimer's disease ELI LILLY AND COMPANY (US) 1996-11-20 EP disclosed
US-5462954-A Antiinflammatory, antiallergens; treating asthma ELI LILLY AND COMPANY (US) 1995-10-31 US disclosed
EP-0544488-A2 Substituted phenyl phenol leukotriene antagonists ELI LILLY AND COMPANY (US) 1993-06-02 EP disclosed