SCHEMBL8567454

SCHEMBL8567454

O=c1ccc2ccc(NC3CCNC3)cc2[nH]1

nearest known ligand 0.48

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ITK Q08881 3/20 0.48
CHEK1 O14757 1/20 0.46
PARP14 Q460N5 1/20 0.43
BRD4 O60885 4/20 0.43
ATAD2 Q6PL18 4/20 0.43
AR P10275 4/20 0.42
KIF11 P52732 1/20 0.42
PRKCQ Q04759 1/20 0.42
AXL P30530 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8264491 0.85 AR (0.51) ITKARKIF11
SCHEMBL4300332 0.83 ITK (0.47) ITKPARP14BRD4ATAD2AR
SCHEMBL1049975 0.81 BRD4 (0.46) ITKCHEK1BRD4ATAD2
SCHEMBL1199874 0.76 KIF11 (0.46) ARKIF11
SCHEMBL23360040 0.76 HTR6 (0.51) ITKBRD4ATAD2
SCHEMBL21460268 0.76 HTR6 (0.51) ITKBRD4ATAD2
SCHEMBL29862859 0.76 HTR6 (0.51) ITKBRD4ATAD2
SCHEMBL21460280 0.74 ITK (0.42) ITKPARP14BRD4ATAD2PRKCQ
SCHEMBL21460246 0.74 PDK2 (0.43) ITKCHEK1PARP14PRKCQAXL
SCHEMBL4292261 0.73 PRKCQ (0.41) ITKCHEK1PARP14BRD4ATAD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5723627-A BACTERICIDES BAYER AKTIENGESELLSCHAFT (DE) 1998-03-03 US disclosed
US-5648493-A MULTISTAGE PROCESS BY CONDENSING AN OXO COMPOUND WITH AN AMINO COMPOUND TO PRODUCE AN IMINE THEN REACTING WITH AN OXO QUINOLINE CARBOXYLIC ACID BAYER AKTIENGESELLSCHAFT (DE) 1997-07-15 US disclosed
US-5061712-A BACTERICIDES BAYER AKTIENGESELLSCHAFT (DE) 1991-10-29 US disclosed