SCHEMBL8568486

SCHEMBL8568486

Cc1cc2c(c(C)c1O)CCC(C)(C)NC2

nearest known ligand 0.31

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.31
PTGS1 P23219 1/20 0.31
PTGS2 P35354 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
TSHR P16473 1/20 0.31
DRD2 P14416 1/20 0.30
DRD1 P21728 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8408660 0.84 HTT (0.33)
SCHEMBL8922080 0.70 MEN1 (0.43) ACHE
SCHEMBL30440069 0.65 CTSB (0.39) PTGS1PTGS2CYP1A2CYP3A4TSHR
SCHEMBL2481913 0.65 CTSB (0.39) PTGS1PTGS2CYP1A2CYP3A4TSHR
SCHEMBL9810709 0.64 CA1 (0.39) ACHEPTGS1PTGS2CYP1A2
SCHEMBL4467796 0.62 ACHE (0.34) ACHEPTGS1PTGS2CYP1A2CYP3A4
SCHEMBL8406862 0.62 ACHE (0.31) ACHEPTGS1PTGS2CYP1A2CYP3A4
SCHEMBL10084011 0.61 PTGS1 (0.41) PTGS1PTGS2CYP1A2CYP3A4TSHR
SCHEMBL8571087 0.61 TSHR (0.32) PTGS1PTGS2CYP1A2CYP3A4TSHR
SCHEMBL19289984 0.61 EGLN1 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0863878-A1 CYCLIC NITRONES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM HOECHST MARION ROUSSEL, INC. (US) 1998-09-16 EP disclosed
WO-1997010218-A1 CYCLIC NITRONES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM HOECHST MARION ROUSSEL, INC. (US) 1997-03-20 WO disclosed