SCHEMBL8568524

SCHEMBL8568524

CCOC(=O)Cc1nsc(NC(=O)OC)n1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.43
MAPK1 P28482 1/20 0.43
SMN1; SMN2 Q16637 4/20 0.41
MAPT P10636 3/20 0.40
LMNA P02545 2/20 0.40
GAA P10253 2/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA9 Q16790 1/20 0.40
KDM4E B2RXH2 1/20 0.40
HTT P42858 1/20 0.40
POLB P06746 1/20 0.39
ALDH1A1 P00352 4/20 0.39
HSD17B10 Q99714 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8567632 0.93 TSHR (0.47) TSHRMAPK1SMN1; SMN2MAPTLMNA
SCHEMBL6761097 0.89 ALDH1A1 (0.43) TSHRMAPK1SMN1; SMN2MAPTLMNA
SCHEMBL8573320 0.88 NPC1 (0.44) TSHRSMN1; SMN2MAPTLMNANPC1
SCHEMBL10840353 0.87 SMN1; SMN2 (0.43) TSHRMAPK1SMN1; SMN2LMNAGAA
SCHEMBL8572990 0.85 KDM4E (0.46) TSHRMAPK1SMN1; SMN2MAPTLMNA
SCHEMBL8572316 0.83 TSHR (0.57) TSHRMAPK1SMN1; SMN2LMNAGAA
SCHEMBL8569581 0.82 ALDH1A1 (0.44) TSHRSMN1; SMN2MAPTLMNANPC1
SCHEMBL8571891 0.81 SMN1; SMN2 (0.53) TSHRMAPK1SMN1; SMN2LMNANPC1
SCHEMBL14647559 0.81 KDM4E (0.52) SMN1; SMN2MAPTLMNAGAANPC1
SCHEMBL6757740 0.81 ALDH1A1 (0.45) SMN1; SMN2MAPTLMNAGAANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5705650-A Process for preparing 1,2,4-thiadiazole derivatives KATAYAMA SEIYAKUSYO CO., LTD. (JP) 1998-01-06 US disclosed
US-5585494-A Process for preparing 1,2,4-thiadiazole derivatives KATAYAMA SEIYAKUSYO CO. LTD. (JP) 1996-12-17 US disclosed
EP-0536900-A2 Process for preparing 1,2,4-Thiadiazole Derivatives KATAYAMA SEIYAKUSYO CO. Ltd. (JP) 1993-04-14 EP disclosed