SCHEMBL8568665

SCHEMBL8568665

CS(=O)(=O)Nc1ccc2c(c1)CCC1(CCNCC1)O2

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.44
HTR6 P50406 1/20 0.40
TRIM24 O15164 1/20 0.40
BRD1 O95696 1/20 0.40
BRPF1 P55201 1/20 0.40
HRH3 Q9Y5N1 2/20 0.39
KCNH2 Q12809 2/20 0.39
MLNR O43193 1/20 0.39
CYP2D6 P10635 1/20 0.39
GHSR Q92847 1/20 0.39
NR3C2 P08235 1/20 0.38
HTR2A P28223 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8565340 0.99 PKM (0.43) PKMHTR6TRIM24BRD1BRPF1
SCHEMBL8913770 0.90 ADRA1D (0.41) KCNH2
SCHEMBL267585 0.79 ADRA1D (0.56) KCNH2
Hydrochloric Acid SCHEMBL8912554 0.79 EPHX2 (0.52) PKMTRIM24BRD1BRPF1HRH3
Hydrochloric Acid SCHEMBL261711 0.78 ADRA1D (0.55) KCNH2
SCHEMBL8914795 0.78 HDAC3 (0.41) KCNH2NR3C2
Hydrochloric Acid SCHEMBL8912935 0.77 HDAC3 (0.41) KCNH2NR3C2
SCHEMBL7849142 0.77 ADRA1D (0.56) KCNH2
Hydrochloric Acid SCHEMBL8912790 0.76 HTR6 (0.37) HTR6MLNRNR3C2HTR2A
SCHEMBL8566857 0.76 ADRA1D (0.47) KCNH2HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0431943-B1 Spiro(pyran)piperidine derivatives MERCK & CO INC (US) 1998-07-15 EP disclosed
EP-0431943-A2 Nitrogen-containing spirocycles MERCK & CO. INC. (US) 1991-06-12 EP disclosed