SCHEMBL8568843

SCHEMBL8568843

Cc1c(C#N)c2n(c1-c1cccnc1)C(F)C(F)C(F)C2

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 7/20 0.42
KDM4E B2RXH2 5/20 0.41
HSD17B10 Q99714 3/20 0.41
HTT P42858 2/20 0.41
TSHR P16473 2/20 0.39
MAPK1 P28482 2/20 0.39
DYRK1A Q13627 2/20 0.39
HPGD P15428 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
CYP11B1 P15538 3/20 0.38
ALDH1A1 P00352 2/20 0.38
MAOA P21397 1/20 0.38
RXFP1 Q9HBX9 1/20 0.37
TP53 P04637 1/20 0.37
CCNC P24863 1/20 0.37
CDK8 P49336 1/20 0.37
CDK19 Q9BWU1 1/20 0.37
ADORA1 P30542 2/20 0.36
ADORA2A P29274 1/20 0.36
AR P10275 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7953590 0.70 CYP11B2 (0.44) CYP11B2KDM4EHSD17B10HTTTSHR
SCHEMBL7590017 0.70 CYP11B2 (0.44) CYP11B2KDM4EHSD17B10HTTTSHR
SCHEMBL7590158 0.65 CYP11B2 (0.56) CYP11B2KDM4EHSD17B10HTTTSHR
SCHEMBL7967494 0.64 CYP11B2 (0.41) CYP11B2KDM4EHSD17B10HTTTSHR
SCHEMBL7961492 0.64 CYP11B2 (0.43) CYP11B2KDM4EHSD17B10HTTTSHR
SCHEMBL5744189 0.62 DYRK1A (0.57) CYP11B2KDM4EHSD17B10HTTTSHR
SCHEMBL3162665 0.61 NTRK1 (0.54) CYP11B2KDM4EHSD17B10HTTDYRK1A
Hydrochloric Acid SCHEMBL5743585 0.61 DYRK1A (0.56) CYP11B2KDM4EHSD17B10HTTTSHR
SCHEMBL7587234 0.60 ABCC1 (0.44) CYP11B2KDM4EHSD17B10HTTTSHR
SCHEMBL23973953 0.60 CYP11B2 (0.47) CYP11B2KDM4EHSD17B10HTTTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0833635-A1 NOVEL USE FOR PYRROLE DERIVATIVES Aventis Pharma S.A. (FR) 1998-04-08 EP disclosed
WO-1997000073-A1 NOVEL USE FOR PYRROLE DERIVATIVES RHONE-POULENC RORER S.A. (FR) 1997-01-03 WO disclosed