SCHEMBL8569558

SCHEMBL8569558

CC(=O)Oc1cccc(C=CC(=O)OC(=O)C=Cc2cccc(OC(C)=O)c2)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCHE P06276 4/20 0.55
KMT2A Q03164 4/20 0.52
KDM4E B2RXH2 3/20 0.52
MEN1 O00255 3/20 0.52
GAA P10253 1/20 0.52
LMNA P02545 3/20 0.51
CYP3A4 P08684 2/20 0.51
IMPDH2 P12268 1/20 0.49
SMN1; SMN2 Q16637 3/20 0.49
ALDH1A1 P00352 1/20 0.49
MAOB P27338 2/20 0.48
FOS P01100 1/20 0.48
JUN P05412 1/20 0.48
MAPT P10636 2/20 0.47
TTR P02766 1/20 0.47
TP53 P04637 1/20 0.47
ACHE P22303 1/20 0.47
NPC1 O15118 2/20 0.47
ALOX5 P09917 1/20 0.47
CYP1A1 P04798 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8569555 1.00 BCHE (0.55) BCHEKMT2AKDM4EMEN1GAA
SCHEMBL8569560 0.96 KMT2A (0.54) BCHEKMT2AKDM4EMEN1GAA
SCHEMBL15996560 0.87 JUN (0.57) BCHEKMT2AKDM4EMEN1GAA
SCHEMBL1711135 0.86 KDM4E (0.66) BCHEKMT2AKDM4EMEN1LMNA
SCHEMBL1711133 0.86 KDM4E (0.66) BCHEKMT2AKDM4EMEN1LMNA
SCHEMBL4713549 0.84 BCHE (0.55) BCHEKMT2AKDM4EMEN1GAA
SCHEMBL4713551 0.84 BCHE (0.55) BCHEKMT2AKDM4EMEN1GAA
SCHEMBL23343707 0.82 CYP3A4 (0.56) BCHEKMT2AKDM4EMEN1LMNA
SCHEMBL716895 0.82 KMT2A (0.60) BCHEKMT2AKDM4EMEN1LMNA
SCHEMBL716894 0.82 KMT2A (0.60) BCHEKMT2AKDM4EMEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0526642-B1 TRITERPENE DERIVATIVE SHIONOGI & CO (JP) 1998-04-01 EP disclosed
US-5248807-A Endothelin antagonists, treatment of cardiovascular disorders SHIONOGI & CO., LTD. (JP) 1993-09-28 US disclosed
EP-0526642-A1 TRITERPENE DERIVATIVE SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 1993-02-10 EP disclosed