SCHEMBL8569560

SCHEMBL8569560

CC(=O)Oc1cccc(C=CC(=O)OC(=O)C=Cc2ccccc2)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.54
BCHE P06276 2/20 0.52
ALOX5 P09917 2/20 0.50
KDM4E B2RXH2 4/20 0.49
MEN1 O00255 2/20 0.49
GAA P10253 1/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
ALDH1A1 P00352 2/20 0.49
PTGS1 P23219 1/20 0.49
PTGS2 P35354 1/20 0.49
MAOB P27338 2/20 0.48
FOS P01100 1/20 0.48
JUN P05412 1/20 0.48
LMNA P02545 2/20 0.48
CYP3A4 P08684 2/20 0.48
TTR P02766 1/20 0.48
TP53 P04637 1/20 0.48
MAPT P10636 1/20 0.48
GLA P06280 1/20 0.47
TDP1 Q9NUW8 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8569558 0.96 BCHE (0.55) KMT2ABCHEALOX5KDM4EMEN1
SCHEMBL8569555 0.96 BCHE (0.55) KMT2ABCHEALOX5KDM4EMEN1
SCHEMBL716895 0.88 KMT2A (0.60) KMT2ABCHEALOX5KDM4EMEN1
SCHEMBL716894 0.88 KMT2A (0.60) KMT2ABCHEALOX5KDM4EMEN1
SCHEMBL1711135 0.85 KDM4E (0.66) KMT2ABCHEALOX5KDM4EMEN1
SCHEMBL1711133 0.85 KDM4E (0.66) KMT2ABCHEALOX5KDM4EMEN1
SCHEMBL15996560 0.83 JUN (0.57) KMT2ABCHEALOX5KDM4EMEN1
SCHEMBL4713551 0.81 BCHE (0.55) KMT2ABCHEALOX5KDM4EMEN1
SCHEMBL4713549 0.81 BCHE (0.55) KMT2ABCHEALOX5KDM4EMEN1
SCHEMBL719415 0.80 KMT2A (0.73) KMT2ABCHEKDM4EMEN1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0526642-B1 TRITERPENE DERIVATIVE SHIONOGI & CO (JP) 1998-04-01 EP disclosed
US-5248807-A Endothelin antagonists, treatment of cardiovascular disorders SHIONOGI & CO., LTD. (JP) 1993-09-28 US disclosed
EP-0526642-A1 TRITERPENE DERIVATIVE SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 1993-02-10 EP disclosed