SCHEMBL8569593

SCHEMBL8569593

CNC(=O)c1cc(F)cc(F)c1C

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.48
HDAC1 Q13547 2/20 0.44
HDAC6 Q9UBN7 2/20 0.44
CES2 O00748 5/20 0.44
CES1 P23141 5/20 0.44
HDAC4 P56524 1/20 0.40
ALDH1A1 P00352 2/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
NUDT1 P36639 1/20 0.35
PARP14 Q460N5 1/20 0.34
PLK1 P53350 2/20 0.34
MAPK14 Q16539 1/20 0.34
IKBKB O14920 1/20 0.33
MAP2K2 P36507 1/20 0.33
MAP2K1 Q02750 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24458098 0.85 GAA (0.44) GAAHDAC1HDAC6CES2CES1
SCHEMBL2062639 0.79 GAA (0.47) GAAHDAC1HDAC6CES2CES1
SCHEMBL19121971 0.79 GAA (0.40) GAAHDAC1HDAC6CES2CES1
SCHEMBL5857864 0.78 CES2 (0.48) HDAC1HDAC6CES2CES1HDAC4
SCHEMBL29657075 0.78 CES2 (0.48) HDAC1HDAC6CES2CES1HDAC4
SCHEMBL16545842 0.78 CES2 (0.48) GAAHDAC1HDAC6CES2CES1
SCHEMBL24571393 0.78 TAS1R3 (0.50) HDAC1HDAC6CES2CES1HDAC4
SCHEMBL8572283 0.77 GAA (0.48) GAAHDAC1HDAC6CES2CES1
SCHEMBL8566781 0.77 GAA (0.44) GAACES2CES1ALDH1A1SMN1; SMN2
SCHEMBL18878112 0.77 CES2 (0.44) GAAHDAC1HDAC6CES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5846990-A Substituted biphenyl isoxazole sulfonamides BRISTOL-MYERS SQUIBB CO. (US) 1998-12-08 US claimed