SCHEMBL8569982

SCHEMBL8569982

N#Cc1c(F)cccc1N1CCCC1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.73
KDM4E B2RXH2 5/20 0.73
HPGD P15428 2/20 0.73
HSD17B10 Q99714 2/20 0.73
L3MBTL1 Q9Y468 3/20 0.65
DRD2 P14416 1/20 0.57
HTR2A P28223 1/20 0.57
HRH1 P35367 1/20 0.57
TDP1 Q9NUW8 1/20 0.49
PDCD1 Q15116 2/20 0.46
CD274 Q9NZQ7 2/20 0.46
AR P10275 1/20 0.44
LMNA P02545 1/20 0.43
GRM2 Q14416 1/20 0.41
GAA P10253 3/20 0.41
NPSR1 Q6W5P4 2/20 0.41
P2RX7 Q99572 1/20 0.40
MAPT P10636 1/20 0.40
TSHR P16473 2/20 0.39
USP2 O75604 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1154557 0.98 KDM4E (0.71) ALDH1A1KDM4EHPGDHSD17B10L3MBTL1
SCHEMBL16793536 0.98 KDM4E (0.71) ALDH1A1KDM4EHPGDHSD17B10L3MBTL1
SCHEMBL29599792 0.85 KDM4E (1.00) ALDH1A1KDM4EHPGDHSD17B10L3MBTL1
SCHEMBL2075341 0.85 ALDH1A1 (0.68) ALDH1A1KDM4EHPGDHSD17B10L3MBTL1
SCHEMBL3076269 0.85 KDM4E (0.68) ALDH1A1KDM4EHPGDHSD17B10L3MBTL1
SCHEMBL10934231 0.85 KDM4E (0.68) ALDH1A1KDM4EHPGDHSD17B10L3MBTL1
SCHEMBL823501 0.85 KDM4E (1.00) ALDH1A1KDM4EHPGDHSD17B10L3MBTL1
SCHEMBL22964425 0.83 KDM4E (0.66) ALDH1A1KDM4EHPGDHSD17B10L3MBTL1
SCHEMBL2072485 0.82 KDM4E (1.00) ALDH1A1KDM4EHPGDHSD17B10L3MBTL1
SCHEMBL1878340 0.81 ALDH1A1 (0.69) ALDH1A1KDM4EHPGDHSD17B10L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0544488-B1 Substituted phenyl phenol leukotriene antagonists LILLY CO ELI (US) 1998-03-11 EP disclosed
CN-1035001-C Substituted phenyl phenol leukotriene antagonists LILLY CO ELI (US) 1997-05-28 CN disclosed
CN-1088906-A The phenyl phenol leukotriene antagonists that replaces LILLY CO ELI (US) 1994-07-06 CN disclosed
EP-0544488-A2 Substituted phenyl phenol leukotriene antagonists ELI LILLY AND COMPANY (US) 1993-06-02 EP disclosed