SCHEMBL8570479

SCHEMBL8570479

c1ccc(C2CCN(c3cccc4c3ncc3cccn34)CC2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHFR P00374 1/20 0.46
GRM2 Q14416 13/20 0.43
KDM4E B2RXH2 2/20 0.43
ALDH1A1 P00352 2/20 0.43
GAA P10253 2/20 0.43
GLA P06280 1/20 0.43
HPGD P15428 1/20 0.43
HSD17B10 Q99714 1/20 0.43
MEN1 O00255 1/20 0.43
NPC1 O15118 1/20 0.43
MAPT P10636 1/20 0.43
MAPK1 P28482 1/20 0.43
RAB9A P51151 1/20 0.43
KMT2A Q03164 1/20 0.43
ATM Q13315 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
SLC6A3 Q01959 2/20 0.41
GRIN2B Q13224 1/20 0.39
HTR2A P28223 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8567794 0.84 ALDH1A1 (0.47) DHFRGRM2KDM4EALDH1A1GAA
SCHEMBL8569163 0.83 GRM2 (0.45) DHFRGRM2SLC6A3CYP2C9CYP2C19
SCHEMBL8569217 0.83 GRM2 (0.44) DHFRGRM2SLC6A3GRIN2BHTR2A
SCHEMBL8569567 0.83 KDM4E (0.47) KDM4EALDH1A1GAAGLAHPGD
SCHEMBL8569974 0.82 ALDH1A1 (0.46) KDM4EALDH1A1GAAGLAHPGD
SCHEMBL8571229 0.80 ALDH1A1 (0.44) KDM4EALDH1A1GAAGLAHPGD
SCHEMBL8568655 0.80 ALDH1A1 (0.44) DHFRKDM4EALDH1A1GAAGLA
SCHEMBL8563754 0.79 HTR3E (0.53) HTR6
SCHEMBL8567573 0.78 ALDH1A1 (0.43) KDM4EALDH1A1GAAGLAHPGD
SCHEMBL8572451 0.76 KDM4E (0.47) KDM4EALDH1A1GAAGLAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0623620-B1 5-HT3 Pyrrolopyrazine derivatives ADIR (FR) 1998-09-09 EP disclosed
US-5599812-A ANTISEROTONINE AGENTS ADIR ET COMPAGNIE (FR) 1997-02-04 US disclosed
EP-0623620-A1 5-HT3 Pyrrolopyrazine derivatives ADIR ET COMPAGNIE (FR) 1994-11-09 EP disclosed