SCHEMBL8570891

SCHEMBL8570891

CCc1nc(N2CCc3ccccc3C2C)nc(O)c1C

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DRD1 P21728 1/20 0.37
PRCP P42785 1/20 0.35
MAPK1 P28482 1/20 0.35
GRM5 P41594 2/20 0.35
HTR1A P08908 2/20 0.33
PRMT5 O14744 2/20 0.33
SPR P35270 3/20 0.33
AKR1C3 P42330 1/20 0.33
LIPE Q05469 1/20 0.33
OPRM1 P35372 1/20 0.33
OPRD1 P41143 1/20 0.33
OPRK1 P41145 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8568770 0.86 DRD1 (0.40) DRD1PRCPMAPK1HTR1APRMT5
SCHEMBL8566400 0.85 DRD1 (0.38) DRD1PRCPMAPK1GRM5SPR
SCHEMBL8567905 0.85 DRD1 (0.38) DRD1PRCPMAPK1GRM5SPR
SCHEMBL8566392 0.85 DRD1 (0.38) DRD1PRCPMAPK1GRM5SPR
SCHEMBL8572994 0.81 GRIN2D (0.39) DRD1PRCPGRM5HTR1APRMT5
SCHEMBL8572844 0.79 SPR (0.41) DRD1MAPK1GRM5SPRAKR1C3
SCHEMBL6989000 0.78 DRD1 (0.39) DRD1PRCPMAPK1HTR1APRMT5
SCHEMBL8572580 0.75 ALDH1A1 (0.36) DRD1GRM5AKR1C3LIPE
Hydrochloric Acid SCHEMBL8568119 0.74 RXFP1 (0.35) OPRM1
SCHEMBL15672478 0.74 DRD1 (0.36) DRD1PRCPMAPK1GRM5SPR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5750531-A ANTISECRETORY AGENTS FOR THE TREATMENT OF PEPTIC ULCER YUHAN CORPORATION (KR) 1998-05-12 US disclosed
EP-0775120-A1 NOVEL PYRIMIDINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF Yuhan Corporation (KR) 1997-05-28 EP disclosed
WO-1996005177-A1 NOVEL PYRIMIDINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF YUHAN CORPORATION (KR) 1996-02-22 WO disclosed