SCHEMBL8573289

SCHEMBL8573289

N#Cc1ccc(C(F)F)c(Cl)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
VCAM1 P19320 1/20 0.41
AR P10275 2/20 0.39
PDK1 Q15118 1/20 0.37
PDK2 Q15119 1/20 0.37
PDK3 Q15120 1/20 0.37
PDK4 Q16654 1/20 0.37
PNMT P11086 1/20 0.35
SLC22A12 Q96S37 1/20 0.35
HSD11B1 P28845 1/20 0.35
EEF2K O00418 1/20 0.35
MAOA P21397 1/20 0.34
MAOB P27338 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
TRPV4 Q9HBA0 1/20 0.34
EGLN2 Q96KS0 2/20 0.34
FLT1 P17948 1/20 0.34
FLT4 P35916 1/20 0.34
KDR P35968 1/20 0.34
CYP11B1 P15538 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18527133 0.84 VCAM1 (0.44) VCAM1ARPDK1PDK2PDK3
SCHEMBL105405 0.80 AR (0.42) VCAM1ARPDK1PDK2PDK3
SCHEMBL8576534 0.78 KIF11 (0.37) PNMTCA2EGLN2CYP11B1CYP11B2
SCHEMBL26620605 0.77 LMNA (0.58) VCAM1ARPDK1PDK2PDK3
SCHEMBL27958799 0.77 AR (0.41) VCAM1ARPDK1PDK2PDK3
SCHEMBL19771883 0.77 AR (0.41) VCAM1ARPDK1PDK2PDK3
SCHEMBL3737426 0.77 PDE2A (0.50) VCAM1ARPDK1PDK2PDK3
SCHEMBL26916884 0.77 LMNA (0.58) VCAM1ARPDK1PDK2PDK3
SCHEMBL9931300 0.76 MEN1 (0.42) PNMTMAOAMAOBCA2EGLN2
SCHEMBL30876218 0.75 GRIN2B (0.39) PNMTCA2EGLN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998016526-A1 TETRAHYDRO-6H-PYRAZINO[1,2-B]ISOQUINOLINE 1,4-DIONES AS APOPROTEIN B-100 INHIBITORS GLAXO GROUP LIMITED (GB) 1998-04-23 WO disclosed