SCHEMBL8573304

SCHEMBL8573304

CNC(=O)c1cccc2[nH]c3ccccc3c12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 2/20 0.56
EGFR P00533 2/20 0.51
SRC P12931 1/20 0.51
KDM4E B2RXH2 1/20 0.50
NPC1 O15118 1/20 0.50
ALDH1A1 P00352 1/20 0.50
LMNA P02545 1/20 0.50
TP53 P04637 1/20 0.50
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 1/20 0.50
MAPT P10636 1/20 0.50
CYP2C9 P11712 1/20 0.50
PKM P14618 1/20 0.50
HPGD P15428 1/20 0.50
TSHR P16473 1/20 0.50
APEX1 P27695 1/20 0.50
CYP2C19 P33261 1/20 0.50
THPO P40225 1/20 0.50
RAB9A P51151 1/20 0.50
PMP22 Q01453 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6007642 0.81 IMPDH2 (0.55) KDM4EALDH1A1LMNAHPGDHSD17B10
SCHEMBL27872217 0.81 IMPDH2 (0.58) KDM4EALDH1A1LMNAMAPTHPGD
SCHEMBL17461856 0.81 MAPT (0.48) PLK1EGFRSRCKDM4ENPC1
SCHEMBL31670359 0.81 NR4A2 (0.55) KDM4EALDH1A1LMNACYP1A2CYP3A4
SCHEMBL30522265 0.81 NR4A2 (0.55) KDM4EALDH1A1LMNACYP1A2CYP3A4
SCHEMBL2181558 0.81 NR4A2 (0.55) KDM4EALDH1A1LMNACYP1A2CYP3A4
SCHEMBL30749415 0.80 PARP1 (0.73) KDM4EALDH1A1LMNACYP1A2MAPT
SCHEMBL2183473 0.80 PARP1 (0.73) KDM4EALDH1A1LMNACYP1A2MAPT
SCHEMBL30455376 0.80 PARP1 (0.73) KDM4EALDH1A1LMNACYP1A2MAPT
SCHEMBL30006934 0.78 IMPDH2 (0.55) KDM4EALDH1A1LMNAHPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014153043-A1 COMPOUNDS AND METHODS FOR TREATING CANCERS HEALTH RESEARCH, INC. (US) 2014-09-25 WO disclosed
CN-1233176-A Substituted tricyclics LILLY CO ELI (US) 1999-10-27 CN disclosed
WO-1998018464-A1 SUBSTITUTED TRICYCLICS ELI LILLY AND COMPANY (US) 1998-05-07 WO disclosed