SCHEMBL8574152

SCHEMBL8574152

CC1Oc2ccc(CC(N)=O)cc2O1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CA2 P00918 1/20 0.43
KDM4E B2RXH2 2/20 0.39
ALDH1A1 P00352 2/20 0.39
LMNA P02545 1/20 0.38
POLB P06746 1/20 0.38
MAPK1 P28482 1/20 0.38
CYP1A2 P05177 2/20 0.37
CYP2C19 P33261 2/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.36
HTR1D P28221 1/20 0.35
HTR1B P28222 1/20 0.35
NPC1 O15118 1/20 0.35
HPGD P15428 1/20 0.35
NFKB1 P19838 1/20 0.35
STAT1 P42224 1/20 0.35
RAB9A P51151 1/20 0.35
NFKB2 Q00653 1/20 0.35
RELA Q04206 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8572275 0.81 HDAC4 (0.37) ALDH1A1LMNAMAPK1CYP1A2CYP2C19
SCHEMBL20051409 0.80 CYP2C9 (0.46) KDM4EALDH1A1LMNAMAPK1CYP2C19
SCHEMBL10274463 0.74 PTGS1 (0.41) ALDH1A1LMNAMAPK1CYP1A2CYP2C19
SCHEMBL8571428 0.74 TSHR (0.53) CA2KDM4EALDH1A1CYP1A2CYP2C19
SCHEMBL11854767 0.74 CYP1A2 (0.36) CYP1A2CYP2C19CYP3A4CYP2C9
SCHEMBL9145627 0.74 PTGS2 (0.46) CA2KDM4EALDH1A1CYP3A4
SCHEMBL3525050 0.72 ALDH1A1 (0.59) CA2KDM4EALDH1A1LMNACYP1A2
SCHEMBL1395778 0.72 CYP3A4 (0.68) ALDH1A1LMNACYP1A2CYP2C19CYP3A4
SCHEMBL28648226 0.72 CYP3A4 (0.46) KDM4EALDH1A1LMNACYP1A2CYP2C19
SCHEMBL10274494 0.72 CNR1 (0.41) KDM4EALDH1A1LMNACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5846990-A Substituted biphenyl isoxazole sulfonamides BRISTOL-MYERS SQUIBB CO. (US) 1998-12-08 US disclosed