SCHEMBL8574170

SCHEMBL8574170

COc1cc2c(c(O)c1OC)C(=O)C(c1ccccc1)(c1cccc(Cl)c1)CO2

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.39
KDM4E B2RXH2 1/20 0.39
TAS2R31 P59538 1/20 0.37
HRH3 Q9Y5N1 1/20 0.35
BACE1 P56817 1/20 0.35
MAPT P10636 3/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
SCN9A Q15858 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.33
ABCB1 P08183 1/20 0.33
ABCG2 Q9UNQ0 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C19 P33261 1/20 0.33
TUBB4A P04350 2/20 0.33
TUBB P07437 2/20 0.33
TUBA3C P0DPH7 2/20 0.33
TUBA1B P68363 2/20 0.33
TUBA4A P68366 2/20 0.33
TUBB4B P68371 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8577398 0.92 GAA (0.38) GAAKDM4EBACE1MAPTSCN9A
SCHEMBL8577388 0.88 GAA (0.39) GAAKDM4ETAS2R31BACE1MAPT
SCHEMBL8575371 0.82 HTR6 (0.42) KDM4EBACE1MAPTABCG2CYP2C19
SCHEMBL8572760 0.82 PLK1 (0.37) BACE1ALDH1A1
SCHEMBL8577569 0.82 ABCG2 (0.42) GAAKDM4ETAS2R31BACE1MAPT
SCHEMBL8576216 0.80 GAA (0.38) GAAKDM4EBACE1MAPTL3MBTL1
SCHEMBL8577389 0.78 GLRA3 (0.34) MAPTNPC1RAB9AMEN1KMT2A
SCHEMBL8572826 0.78 CYP19A1 (0.37) MAPTCYP1A2CYP2C19MEN1KMT2A
SCHEMBL8575417 0.71 RIPK1 (0.41) GAAKDM4ETAS2R31MAPTNPC1
SCHEMBL8577523 0.69 ABCG2 (0.42) GAAKDM4ETAS2R31MAPTNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998017662-A1 PHENYL-SUBSTITUTED BICYCLIC HETEROCYCLYL DERIVATIVES AND THEIR USE NOVARTIS AG (CH) 1998-04-30 WO claimed
WO-1998017662-A1 PHENYL-SUBSTITUTED BICYCLIC HETEROCYCLYL DERIVATIVES AND THEIR USE NOVARTIS AG (CH) 1998-04-30 WO disclosed