SCHEMBL8574371

SCHEMBL8574371

COc1cc(O)c2c(=O)c(-c3cccc(Cl)c3)c[nH]c2c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 7/20 1.00
SRC P12931 1/20 0.76
ABL1 P00519 1/20 0.47
ABL2 P42684 1/20 0.47
PRKAB2 O43741 1/20 0.42
PRKAG1 P54619 1/20 0.42
PRKAA2 P54646 1/20 0.42
PRKAA1 Q13131 1/20 0.42
PRKAG3 Q9UGI9 1/20 0.42
PRKAG2 Q9UGJ0 1/20 0.42
PRKAB1 Q9Y478 1/20 0.42
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41
NPC1 O15118 2/20 0.40
CYP2C9 P11712 2/20 0.40
CYP2C19 P33261 2/20 0.40
MEN1 O00255 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
NFKB1 P19838 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4359046 0.89 EGFR (0.80) EGFRSRCALDH1A1LMNANPC1
SCHEMBL8574541 0.87 EGFR (1.00) EGFRSRCABL1ABL2ALDH1A1
SCHEMBL4358045 0.86 EGFR (0.76) EGFRSRCALDH1A1LMNANPC1
SCHEMBL4361477 0.85 EGFR (0.73) EGFRSRCPRKAB2PRKAG1PRKAA2
SCHEMBL7256744 0.83 EGFR (0.70) EGFRSRCPRKAB2PRKAG1PRKAA2
SCHEMBL4353399 0.80 EGFR (0.66) EGFRSRCABL1ABL2ALDH1A1
SCHEMBL8575803 0.79 EGFR (0.73) EGFRSRCABL1ABL2MEN1
SCHEMBL8576451 0.76 EGFR (1.00) EGFRSRCABL1ABL2NPC1
SCHEMBL8578711 0.75 EGFR (0.78) EGFRSRCABL1ABL2ALDH1A1
SCHEMBL8577298 0.73 EGFR (0.78) EGFRSRCABL1ABL2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998017662-A1 PHENYL-SUBSTITUTED BICYCLIC HETEROCYCLYL DERIVATIVES AND THEIR USE NOVARTIS AG (CH) 1998-04-30 WO claimed
WO-1998017662-A1 PHENYL-SUBSTITUTED BICYCLIC HETEROCYCLYL DERIVATIVES AND THEIR USE NOVARTIS AG (CH) 1998-04-30 WO disclosed