SCHEMBL8574646

SCHEMBL8574646

CC(C)[C@H](NC(=O)OC(C)(C)C)C(=O)OC1CC(=O)NC1=O

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CTSK P43235 2/20 0.40
CTSS P25774 1/20 0.40
PREP P48147 1/20 0.39
CTSL P07711 2/20 0.38
TRPA1 O75762 2/20 0.38
CTSB P07858 1/20 0.38
CA2 P00918 2/20 0.37
CA1 P00915 1/20 0.37
CA7 P43166 1/20 0.37
GAA P10253 1/20 0.36
ELANE P08246 1/20 0.35
KLK5 Q9Y337 1/20 0.35
IDO1 P14902 1/20 0.35
EPHX2 P34913 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
SRC P12931 1/20 0.34
CYP2D6 P10635 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10627589 0.91 CTSL (0.35) CTSKCTSSPREPCTSLTRPA1
SCHEMBL10633587 0.87 EPHX2 (0.42) CTSLCA2CA1CA7GAA
SCHEMBL8576306 0.87 EPHX2 (0.42) CTSLCA2CA1CA7GAA
SCHEMBL9781378 0.83 KMT2A (0.40) GAAIDO1EPHX2KMT2A
SCHEMBL8577285 0.82 CTSL (0.46) CTSKCTSSCTSLCTSBCA2
SCHEMBL10631067 0.82 CTSL (0.46) CTSKCTSSCTSLCTSBCA2
SCHEMBL8695509 0.81 IDO1 (0.41) CTSKCTSSCTSLGAAKLK5
SCHEMBL9228941 0.80 IDO1 (0.40) CTSKCTSSCTSLCTSBGAA
SCHEMBL6741998 0.80 CTSK (0.42) CTSKCTSSPREPCTSLTRPA1
SCHEMBL13869102 0.76 CTSK (0.44) CTSKCTSSPREPCTSLTRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5789386-A WATER SOLUBLE ANTITUMOR AGENTS; INJECTABLE ZAIDAN HOJIN BISEIBUTSU KAGAKU KENKYU KAI (JP) 1998-08-04 US disclosed
EP-0374097-A2 Use of peptide isosteres as retroviral protease inhibitors CIBA-GEIGY AG (CH) 1990-06-20 EP disclosed
EP-0374098-A2 Inhibitors of retroviral proteases CIBA-GEIGY AG (CH) 1990-06-20 EP disclosed
EP-0295316-A2 Antitumor amino acid and peptide derivatives of 1,4-bis[ (aminoalkyl and hydroxyaminoalkyl)- amino]-5,8 dihydroxyanthraquinones AMERICAN CYANAMID COMPANY (US) 1988-12-21 EP disclosed
US-4732970-A Antitumor amino acid and peptide derivatives of 1,4-bis(aminoalkyl and hydroxy-aminoalkyl)amino)-5,8-dihydroxyanthraquinones AMERICAN CYANAMID COMPANY (US) 1988-03-22 US disclosed