SCHEMBL8575658

SCHEMBL8575658

CCCC[Si](CCCC)(CCCC)O[C@@H]1CC(CN2C(=O)c3ccccc3C2=O)N(C(=O)OC(C)(C)C)C1

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 1/20 0.38
SRC P12931 8/20 0.35
PARP1 P09874 2/20 0.35
BRD4 O60885 2/20 0.35
IDO1 P14902 2/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
KLK7 P49862 4/20 0.33
KLK5 Q9Y337 4/20 0.33
PRSS1 P07477 2/20 0.33
PRSS2 P07478 2/20 0.33
PRSS3 P35030 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21286395 0.85 ABCB1 (0.38) ABCB1SRCPARP1BRD4IDO1
SCHEMBL29985450 0.85 ABCB1 (0.38) ABCB1SRCPARP1BRD4IDO1
SCHEMBL3948504 0.85 ABCB1 (0.38) ABCB1SRCPARP1BRD4IDO1
SCHEMBL8568862 0.80 NR1H2 (0.39) ABCB1SRCPARP1MEN1KMT2A
SCHEMBL8568867 0.80 NR1H2 (0.39) ABCB1SRCPARP1MEN1KMT2A
SCHEMBL3952747 0.80 BRD4 (0.39) ABCB1SRCBRD4
SCHEMBL7807928 0.80 BRD4 (0.39) ABCB1SRCBRD4
SCHEMBL19674208 0.79 HSD17B10 (0.40) SRCBRD4IDO1MEN1KMT2A
SCHEMBL8572979 0.79 CYP1A2 (0.43) SRCBRD4IDO1MEN1KMT2A
SCHEMBL3947235 0.79 CYP1A2 (0.43) SRCBRD4IDO1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5726182-A TREATMENT OF BACTERIAL INFECTIONS ABBOTT LABORATORIES (US) 1998-03-10 US disclosed
US-5599816-A BACTERICIDE ABBOTT LABORATORIES (US) 1997-02-04 US disclosed
WO-1996039407-A1 QUINOLIZINONE TYPE COMPOUNDS ABBOTT LABORATORIES (US) 1996-12-12 WO disclosed