SCHEMBL8575945

SCHEMBL8575945

COC(=O)CCNS(=O)(=O)c1ccc(C)cc1

nearest known ligand 0.63

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.63
ALDH1A1 P00352 12/20 0.61
USP2 O75604 1/20 0.61
LMNA P02545 3/20 0.59
HTT P42858 2/20 0.59
HPGD P15428 1/20 0.59
MEN1 O00255 2/20 0.57
KMT2A Q03164 2/20 0.57
GAA P10253 2/20 0.56
KDM4E B2RXH2 2/20 0.56
GLA P06280 1/20 0.56
L3MBTL1 Q9Y468 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28399402 0.91 ALDH1A1 (0.65) MAPTALDH1A1USP2LMNAHTT
SCHEMBL19078974 0.88 ALDH1A1 (0.69) MAPTALDH1A1LMNAHTT
SCHEMBL13223680 0.88 ALDH1A1 (0.69) MAPTALDH1A1LMNAHTT
SCHEMBL12207107 0.86 CA12 (0.61) MAPTALDH1A1LMNAHPGDMEN1
SCHEMBL18498935 0.86 IDO1 (0.56) ALDH1A1HPGDMEN1KMT2AGAA
SCHEMBL9464524 0.85 CA12 (0.61) MAPTALDH1A1LMNAGAAKDM4E
SCHEMBL8576412 0.85 ALDH1A1 (0.56) MAPTALDH1A1USP2LMNAHTT
SCHEMBL3103190 0.84 MEP1B (0.67) MAPTALDH1A1LMNAHPGDKMT2A
SCHEMBL4541169 0.83 ALDH1A1 (0.73) MAPTALDH1A1USP2LMNAHTT
SCHEMBL15869133 0.83 ALDH1A1 (0.64) MAPTALDH1A1USP2LMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10385055-B2 Tricyclic gyrase inhibitors MERCK SHARP & DOHME CORP. (US) 2019-08-20 US disclosed
US-5783699-A MAY BE CONJUGATED TO ANTIGENS, HAPTENS, ANTIBODIES IN IMMUNOASSAYS ABBOTT LABORATORIES (US) 1998-07-21 US disclosed
US-5669819-A IMMUNOASSAY ABBOTT LABORATORIES (US) 1997-09-23 US disclosed
US-5565570-A REACTING AMINE WITH SULFONYL HALIDE IN INERT SOLVENT IN PRESENCE OF BASE TO FORM METAL SALT OF SULFONAMIDE, ACYLATING WITH ACTIVATED PHENANTHRIDINE-6-CARBOXYLIC ACID TO FORM CHEMILUMINESCENT SALT ABBOTT LABORATORIES (US) 1996-10-15 US disclosed
US-5545739-A E.G., 5-METHYL-6-(N-2-CARBOXYETHYL-N=(2-CARBOXYETHYL)-PHENANTHRIDIN IUMCARBOXAMIDE CHLORIDE; IMMUNOASSAYS; STABILITY; SENSITIVITY ABBOTT LABORATORIES (US) 1996-08-13 US disclosed
US-5543524-A FORMING A SULFONAMIDE FROM AND AMINE AND A SULFONYL HALIDE AND AND ACYLATING WITH A CARBONYL HALIDE OF AN ACTIVATED ACRIDINE SALT ABBOTT LABORATORIES (US) 1996-08-06 US disclosed
US-5468646-A Chemiluminescent acridinium salts ABBOTT LABORATORIES (US) 1995-11-21 US disclosed
EP-0273115-B1 Chemiluminescent acridinium and phenanthridinium salts ABBOTT LAB (US) 1994-09-07 EP disclosed
EP-0273115-A2 Chemiluminescent acridinium and phenanthridinium salts ABBOTT LABORATORIES (US) 1988-07-06 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10385055-B2 Tricyclic gyrase inhibitors TOP1, TOP2A, TOP2B MAPT 2765/4885ALDH1A1 1898/4885USP2 2671/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.