SCHEMBL8576705

SCHEMBL8576705

COC(=O)C1CN(C(=O)OC(C)(C)C)CCN1Cc1cccc2ccccc12

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.52
HTT P42858 1/20 0.45
KMT2A Q03164 1/20 0.43
TMEM97 Q5BJF2 2/20 0.42
SIGMAR1 Q99720 2/20 0.42
FAAH O00519 1/20 0.42
BACE1 P56817 1/20 0.42
CHRM2 P08172 1/20 0.41
CHRM4 P08173 1/20 0.41
CHRM1 P11229 1/20 0.41
CHRM3 P20309 1/20 0.41
GPR119 Q8TDV5 3/20 0.41
MC4R P32245 2/20 0.41
MC1R Q01726 2/20 0.41
MC3R P41968 1/20 0.41
GRM2 Q14416 1/20 0.40
GRM3 Q14832 1/20 0.40
NR1H2 P55055 1/20 0.39
NR1H3 Q13133 1/20 0.39
DTYMK P23919 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30867751 0.83 GPR119 (0.50) ACHEGPR119KDM4E
SCHEMBL17913813 0.83 GPR119 (0.50) ACHEGPR119KDM4E
SCHEMBL23293544 0.79 ACHE (0.60) ACHEKMT2AFAAHCHRM2CHRM4
SCHEMBL30422174 0.79 ACHE (0.60) ACHEKMT2AFAAHCHRM2CHRM4
SCHEMBL16830462 0.79 ACHE (0.60) ACHEKMT2AFAAHCHRM2CHRM4
SCHEMBL4573479 0.79 P2RX7 (0.46) ACHEHTTKMT2AGPR119
SCHEMBL30763175 0.78 GPR119 (0.48) GPR119
SCHEMBL22800954 0.77 CYP3A4 (0.47) HTTKMT2AGPR119KDM4E
SCHEMBL1014461 0.75 ACHE (0.45) ACHEKMT2ABACE1KDM4EAPOBEC3A
SCHEMBL10181653 0.74 PDE4B (0.44) KMT2AGPR119NR1H2NR1H3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5736539-A ANITCARCINOGENIC AGENTS MERCK & CO., INC. (US) 1998-04-07 US disclosed
WO-1995000497-A1 INHIBITORS OF FARNESYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 1995-01-05 WO disclosed