SCHEMBL8577158

SCHEMBL8577158

[CH2]C(O)[CH]Cc1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAOB P27338 1/20 0.48
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
ARG2 P78540 1/20 0.42
TSHR P16473 1/20 0.39
CALM1 P0DP23 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
CYP1A2 P05177 1/20 0.35
TRPA1 O75762 2/20 0.35
TOP1 P11387 1/20 0.35
IDO1 P14902 3/20 0.34
THRB P10828 1/20 0.34
CES2 O00748 1/20 0.34
CES1 P23141 1/20 0.34
AKR1B1 P15121 1/20 0.34
EPHX1 P07099 1/20 0.34
NOS3 P29474 1/20 0.34
NOS1 P29475 1/20 0.34
NOS2 P35228 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4155331 0.82 MAOB (0.48) MAOBCA1CA2ARG2TSHR
SCHEMBL3295095 0.82 MAOB (0.48) MAOBCA1CA2ARG2TSHR
SCHEMBL8174260 0.77 MAOB (0.48) MAOBCA1CA2ARG2TRPA1
SCHEMBL10755711 0.76 MAOB (0.46) MAOBCA1CA2ARG2TSHR
SCHEMBL8666884 0.74 CYP1A2 (0.47) MAOBCA1CA2ARG2CYP1A2
SCHEMBL5347335 0.74 MAOB (0.44) MAOBCA1CA2ARG2TSHR
SCHEMBL3295725 0.74 TRPA1 (0.46) MAOBCA1CA2ARG2TRPA1
SCHEMBL1289345 0.71 MAOB (0.52) MAOBCA1CA2ARG2CALM1
SCHEMBL11098509 0.71 SIGMAR1 (0.50) MAOBTRPA1EPHX1
SCHEMBL5680524 0.71 MAOB (0.46) MAOBTRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5776933-A Method of inhibiting protease E. R. SQUIBB & SONS, INC. (US) 1998-07-07 US disclosed
US-5760036-A ENZYME INHIBITORS OF RETROVIRAL PROTEASE FOR PREVENTION OF AIDS E. R. SQUIBB & SONS, INC. (US) 1998-06-02 US disclosed