SCHEMBL8577299

SCHEMBL8577299

C#Cc1cc(Br)ccc1C(=O)O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.48
GLA P06280 1/20 0.48
AKR1C3 P42330 2/20 0.42
MYC P01106 1/20 0.41
NR4A1 P22736 1/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
RXFP1 Q9HBX9 1/20 0.40
GRIN1 Q05586 1/20 0.40
GRIN2A Q12879 1/20 0.40
GRIN2B Q13224 1/20 0.40
GRIN2C Q14957 1/20 0.40
GPR35 Q9HC97 1/20 0.40
ACLY P53396 1/20 0.40
APEX1 P27695 1/20 0.39
DGAT1 O75907 1/20 0.39
SRD5A1 P18405 1/20 0.39
SRD5A2 P31213 1/20 0.39
CYP1A2 P05177 2/20 0.38
CES2 O00748 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Benzene SCHEMBL28354519 0.83 KDM4E (0.52) KDM4EGLAAKR1C3MYCNR4A1
SCHEMBL257347 0.81 KDM4E (0.48) KDM4EGLAMYCNR4A1MEN1
SCHEMBL5667262 0.80 ACMSD (0.46) KDM4EMEN1KMT2ARXFP1CYP1A2
SCHEMBL26732932 0.79 NR4A2 (0.48) KDM4EGLACYP1A2CYP2C9HPGD
SCHEMBL1713016 0.78 KDM4E (0.47) KDM4EMYCSRD5A2CYP1A2
SCHEMBL689510 0.78 CYP1A2 (0.39) KDM4EMEN1KMT2ACYP1A2ALOX15
SCHEMBL8573798 0.77 CSNK2A1 (0.50) KDM4EAKR1C3MEN1KMT2AACLY
SCHEMBL8576509 0.77 SMN1; SMN2 (0.57) KDM4EMYCNR4A1MEN1KMT2A
Hydrochloric Acid SCHEMBL3453575 0.77 KDM4E (0.46) KDM4EMYCSRD5A2CYP1A2
SCHEMBL4037266 0.77 KDM4E (0.55) KDM4EGLAMEN1KMT2ARXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1068587-C Ortho-substituted benzoic acid derivatives MERCK PATENT GMBH (DE) 2001-07-18 CN disclosed
US-5849796-A Ortho-substituted benzoil acid derivatives MERCK PATENT GELSELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1998-12-15 US disclosed
CN-1125722-A Ortho-substituted benzoic acid derivatives MERCK PATENT GMBH (DE) 1996-07-03 CN disclosed