SCHEMBL8577613

SCHEMBL8577613

O=C(CBr)c1cnc(C(F)F)nc1Cl

nearest known ligand 0.33

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 1/20 0.33
GSK3B P49841 1/20 0.33
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
P2RX7 Q99572 2/20 0.30
KEAP1 Q14145 1/20 0.30
NFE2L2 Q16236 1/20 0.30
JUN P05412 1/20 0.30
NFKB1 P19838 1/20 0.30
NFKB2 Q00653 1/20 0.30
RELA Q04206 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8566570 0.82 TSHR (0.36) KDM4EALDH1A1
SCHEMBL8558079 0.79 POLB (0.35) KDM4EALDH1A1KEAP1NFE2L2JUN
SCHEMBL8566197 0.75 NFKB1 (0.35) KEAP1NFE2L2JUNNFKB1NFKB2
SCHEMBL8560094 0.74 P2RX7 (0.36) P2RX7
SCHEMBL8565949 0.73 NR4A1 (0.41) ALDH1A1
SCHEMBL26598773 0.69
SCHEMBL8176734 0.69 POLB (0.36)
SCHEMBL30843825 0.68 GSK3B (0.37) PTPN1GSK3BP2RX7
SCHEMBL8566402 0.65 APLNR (0.33)
SCHEMBL3921448 0.65 GSK3B (0.41) PTPN1GSK3BALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5773388-A Pyrimidine derivatives, herbicides and plant growth regulators NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 1998-06-30 US disclosed
EP-0713872-A1 NOVEL PYRIMIDINE DERIVATIVE, HERBICIDE AND PLANT GROWTH REGULATOR NISSAN CHEMICAL INDUSTRIES, LIMITED (JP) 1996-05-29 EP disclosed