SCHEMBL8577947

SCHEMBL8577947

N[C@@H](CO)Cc1ccccc1C(=O)Nc1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.60

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
P2RX1 P51575 15/20 0.60
P2RX7 Q99572 4/20 0.57
P2RX4 Q99571 3/20 0.57
TMPRSS4 Q9NRS4 3/20 0.53
P2RX3 P56373 1/20 0.51
MAPT P10636 1/20 0.50
THRB P10828 1/20 0.50
PTGS1 P23219 1/20 0.48
RXFP1 Q9HBX9 1/20 0.46
NFKB1 P19838 1/20 0.46
NFKB2 Q00653 1/20 0.46
RELA Q04206 1/20 0.46
TACR1 P25103 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8720167 0.81 BCAT2 (0.57)
SCHEMBL8577008 0.78 P2RX1 (0.49) P2RX1P2RX7P2RX4TMPRSS4P2RX3
SCHEMBL8580261 0.77 NPC1 (0.50) MAPTPTGS1NFKB1NFKB2RELA
SCHEMBL8576416 0.76 P2RX1 (0.42) P2RX1P2RX7P2RX4TMPRSS4P2RX3
SCHEMBL5666099 0.75 P2RX1 (1.00) P2RX1P2RX7P2RX4TMPRSS4P2RX3
Hydrochloric Acid SCHEMBL8717918 0.74 HTT (0.52) RXFP1
SCHEMBL10797383 0.74 P2RX1 (0.73) P2RX1P2RX7P2RX4TMPRSS4P2RX3
SCHEMBL127962 0.74 P2RX1 (1.00) P2RX1P2RX7P2RX4TMPRSS4P2RX3
SCHEMBL9081796 0.74 GAA (0.45)
SCHEMBL28258728 0.73 P2RX1 (1.00) P2RX1P2RX7P2RX4TMPRSS4P2RX3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998017636-A1 PHENYLALANINOL DERIVATIVES FOR THE TREATMENT OF CENTRAL NERVOUS SYSTEM DISORDERS ORTHO PHARMACEUTICAL CORPORATION (US) 1998-04-30 WO disclosed