SCHEMBL8580261

SCHEMBL8580261

N[C@@H](CO)Cc1ccccc1C(=O)Nc1ccc(Cl)c(Cl)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.50
RAB9A P51151 4/20 0.50
KDR P35968 3/20 0.50
FLT1 P17948 2/20 0.50
SMO Q99835 1/20 0.47
FPR2 P25090 1/20 0.47
GRM4 Q14833 1/20 0.47
KMT2A Q03164 4/20 0.46
MEN1 O00255 3/20 0.46
MAPK14 Q16539 2/20 0.46
FADS1 O60427 1/20 0.46
PTGS1 P23219 2/20 0.46
TBXAS1 P24557 1/20 0.46
MAPK1 P28482 1/20 0.46
PTGS2 P35354 1/20 0.46
MAPT P10636 3/20 0.46
KDM4E B2RXH2 2/20 0.46
PKM P14618 1/20 0.46
MAOB P27338 1/20 0.45
CASP3 P42574 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8720167 0.82 BCAT2 (0.57) NPC1RAB9ASMOKMT2AMEN1
SCHEMBL8575106 0.81 NPC1 (0.50) NPC1RAB9AKDRFLT1SMO
SCHEMBL8577947 0.77 P2RX1 (0.60) PTGS1MAPTNFKB1NFKB2RELA
SCHEMBL4254011 0.75 RAB9A (0.68) NPC1RAB9ASMOGRM4KMT2A
SCHEMBL9081796 0.74 GAA (0.45) KDM4EALDH1A1
SCHEMBL1963713 0.74 FADS1 (0.76) NPC1RAB9AGRM4KMT2AMEN1
Hydrochloric Acid SCHEMBL8720439 0.73 GAA (0.44) KDM4EALDH1A1CA2
SCHEMBL10489740 0.73 NPC1 (0.69) NPC1RAB9AGRM4KMT2AMEN1
SCHEMBL28093056 0.73 PTGS1 (0.72) NPC1RAB9AGRM4KMT2AMEN1
Hydrochloric Acid SCHEMBL8717918 0.72 HTT (0.52) NPC1RAB9AKMT2AMEN1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998017636-A1 PHENYLALANINOL DERIVATIVES FOR THE TREATMENT OF CENTRAL NERVOUS SYSTEM DISORDERS ORTHO PHARMACEUTICAL CORPORATION (US) 1998-04-30 WO disclosed