SCHEMBL8577987

SCHEMBL8577987

CCCn1c(=O)c2c(nc(C3CCCC3)n2Cc2ccccc2)n(C(C)c2ccc(C(=O)OC)cc2)c1=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 6/20 0.45
ADORA2A P29274 4/20 0.43
ADORA2B P29275 3/20 0.43
MAPT P10636 2/20 0.41
ADORA1 P30542 4/20 0.41
KMT2A Q03164 1/20 0.41
ALDH1A1 P00352 2/20 0.40
KDM4E B2RXH2 1/20 0.40
PKM P14618 1/20 0.40
PDE5A O76074 2/20 0.40
P2RX3 P56373 1/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
TSHR P16473 2/20 0.38
LMNA P02545 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
TP53 P04637 1/20 0.38
MAPK1 P28482 1/20 0.38
HSD17B10 Q99714 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8577988 0.86 ADORA3 (0.51) ADORA3ADORA2AADORA2BADORA1KMT2A
SCHEMBL8579260 0.78 ADORA3 (0.56) ADORA3ADORA2AADORA2BADORA1KMT2A
SCHEMBL8579493 0.77 ADORA3 (0.60) ADORA3ADORA2AADORA2BADORA1KMT2A
SCHEMBL8577867 0.77 ADORA3 (0.57) ADORA3ADORA2AADORA2BADORA1KMT2A
SCHEMBL8576493 0.77 ADORA2A (0.59) ADORA3ADORA2AADORA2BADORA1KMT2A
SCHEMBL8581790 0.76 ADORA3 (0.56) ADORA3ADORA2AADORA2BADORA1KMT2A
SCHEMBL8577877 0.76 ADORA2B (0.60) ADORA3ADORA2AADORA2BADORA1KMT2A
SCHEMBL8576951 0.76 ADORA3 (0.61) ADORA3ADORA2AADORA2BADORA1KMT2A
SCHEMBL8576968 0.76 ADORA3 (0.56) ADORA3ADORA2AADORA2BADORA1KMT2A
SCHEMBL8576828 0.76 ADORA3 (0.57) ADORA3ADORA2AADORA2BADORA1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5719279-A CHOLINOMIMETICS BOEHRINGER INGELHEIM KG (DE) 1998-02-17 US disclosed
WO-1994003456-A1 ASYMMETRICALLY SUBSTITUTED XANTHINE WITH ADENOSINE-ANTAGONISTIC PROPERTIES BOEHRINGER INGELHEIM KG (DE) 1994-02-17 WO disclosed