SCHEMBL8578367

SCHEMBL8578367

COc1ccc2c(c1)c(C(Cc1ccccc1)C(=O)O)c(C)n2C(=O)c1ccccc1

nearest known ligand 0.61

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.61
CYP1A2 P05177 1/20 0.61
CYP2D6 P10635 1/20 0.61
CYP2C9 P11712 1/20 0.61
TSHR P16473 1/20 0.61
NFKB1 P19838 1/20 0.61
HIF1A Q16665 1/20 0.61
NPSR1 Q6W5P4 1/20 0.61
PLA2G2A P14555 1/20 0.59
PTGS2 P35354 9/20 0.56
AKR1C3 P42330 5/20 0.53
AKR1C2 P52895 5/20 0.53
AKR1C4 P17516 1/20 0.53
AKR1C1 Q04828 1/20 0.53
PPARG P37231 2/20 0.53
PTGS1 P23219 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6423697 0.83 PTGS2 (0.54) LMNACYP1A2CYP2D6CYP2C9TSHR
SCHEMBL15658049 0.81 PTGS2 (0.66) LMNACYP1A2CYP2D6CYP2C9HIF1A
SCHEMBL11553568 0.81 PTGS2 (0.65) LMNACYP1A2CYP2D6CYP2C9HIF1A
SCHEMBL6102634 0.80 PTGS2 (0.43) LMNACYP1A2CYP2D6CYP2C9TSHR
SCHEMBL6458883 0.80 PTGS2 (0.65) LMNACYP1A2CYP2D6CYP2C9HIF1A
SCHEMBL10909068 0.80 LMNA (0.59) LMNACYP1A2CYP2D6CYP2C9TSHR
SCHEMBL8430489 0.80 PTGS2 (0.67) LMNACYP1A2CYP2D6CYP2C9HIF1A
SCHEMBL11832986 0.79 PTGS2 (0.63) LMNACYP1A2CYP2D6CYP2C9HIF1A
SCHEMBL6423750 0.79 AKR1C3 (0.53) LMNACYP1A2CYP2D6CYP2C9TSHR
SCHEMBL6425916 0.79 PTGS2 (0.61) NPSR1PTGS2AKR1C3AKR1C2PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5721347-A Esters and amides of substituted pyrrole acetic acids CELL PATHWAYS, INC. (US) 1998-02-24 US disclosed
EP-0485157-A2 Esters and amides of substituted pyrrole acetic acids FGN, INC. (US) 1992-05-13 EP disclosed