SCHEMBL8580408

SCHEMBL8580408

Cc1cc(C=C2SCC(=O)N2N(C)C)cc(C(C)(C)C)c1O

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.41
CYP2C9 P11712 1/20 0.41
PTGS1 P23219 6/20 0.40
PTGS2 P35354 6/20 0.40
EEF2K O00418 1/20 0.39
SRC P12931 1/20 0.39
ALOX5 P09917 2/20 0.39
GAA P10253 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8582463 0.93 CYP1A2 (0.48) CYP1A2CYP2C9PTGS1PTGS2EEF2K
SCHEMBL8585372 0.82 CYP1A2 (0.45) CYP1A2CYP2C9PTGS1PTGS2EEF2K
SCHEMBL8583985 0.81 CYP1A2 (0.47) CYP1A2CYP2C9PTGS1PTGS2EEF2K
SCHEMBL8583892 0.79 CYP1A2 (0.41) CYP1A2CYP2C9PTGS1PTGS2EEF2K
SCHEMBL8580319 0.78 CYP1A2 (0.41) CYP1A2CYP2C9PTGS1PTGS2EEF2K
SCHEMBL8578798 0.76 CYP1A2 (0.51) CYP1A2CYP2C9PTGS1PTGS2EEF2K
SCHEMBL8992131 0.76 PTGS2 (0.48) PTGS1PTGS2ALOX5GAA
SCHEMBL8895623 0.76 PTGS2 (0.48) PTGS1PTGS2ALOX5GAA
SCHEMBL8582530 0.76 CYP1A2 (0.48) CYP1A2CYP2C9PTGS1PTGS2EEF2K
SCHEMBL8580683 0.75 ALDH1A1 (0.40) CYP1A2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5731336-A USING ARYL-SUBSTITUTED RHODAMINES ELI LILLY AND COMPANY (US) 1998-03-24 US disclosed