SCHEMBL8580683

SCHEMBL8580683

CN(C)N1C(=O)CSC1=CCc1cc(C(C)(C)C)c(O)c(C(C)(C)C)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.40
GAA P10253 4/20 0.40
TSHR P16473 3/20 0.40
LMNA P02545 2/20 0.40
TDP1 Q9NUW8 2/20 0.39
MAPT P10636 4/20 0.38
MAPK1 P28482 2/20 0.38
MEN1 O00255 1/20 0.38
USP2 O75604 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
BLM P54132 1/20 0.38
KMT2A Q03164 1/20 0.38
ATM Q13315 1/20 0.38
HIF1A Q16665 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
KDM4E B2RXH2 5/20 0.36
HPGD P15428 2/20 0.35
HTT P42858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8580713 0.84 ALDH1A1 (0.42) ALDH1A1GAATSHRLMNATDP1
SCHEMBL8582463 0.81 CYP1A2 (0.48) ALDH1A1GAAMEN1CYP1A2KMT2A
SCHEMBL8992161 0.75 ALDH1A1 (0.40) ALDH1A1GAATSHRLMNATDP1
SCHEMBL9028884 0.75 ALDH1A1 (0.40) ALDH1A1GAATSHRLMNATDP1
SCHEMBL8580408 0.75 CYP1A2 (0.41) GAACYP1A2
SCHEMBL9029562 0.74 ALDH1A1 (0.40) ALDH1A1GAATSHRLMNATDP1
SCHEMBL8585372 0.74 CYP1A2 (0.45) ALDH1A1GAAMEN1CYP1A2KMT2A
SCHEMBL8933379 0.74 ALDH1A1 (0.40) ALDH1A1GAATSHRLMNATDP1
SCHEMBL8910093 0.72 LMNA (0.37) ALDH1A1GAATSHRLMNATDP1
SCHEMBL8583985 0.71 CYP1A2 (0.47) CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5731336-A USING ARYL-SUBSTITUTED RHODAMINES ELI LILLY AND COMPANY (US) 1998-03-24 US disclosed