SCHEMBL8580439

SCHEMBL8580439

NC(=O)c1cccc(C(N)=O)c1[CH]c1c(C(N)=O)cccc1C(N)=O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.50
KDM4E B2RXH2 3/20 0.50
HPGD P15428 3/20 0.50
MAPT P10636 2/20 0.50
TSHR P16473 1/20 0.50
HSD17B10 Q99714 1/20 0.50
BCAT2 O15382 1/20 0.50
METAP2 P50579 1/20 0.46
GAA P10253 1/20 0.45
PARP1 P09874 5/20 0.44
KEAP1 Q14145 1/20 0.44
NFE2L2 Q16236 1/20 0.44
PDPK1 O15530 1/20 0.44
AURKA O14965 2/20 0.41
LMNA P02545 1/20 0.41
PLK4 O00444 1/20 0.41
CHEK1 O14757 1/20 0.41
DAPK3 O43293 1/20 0.41
MAP4K4 O95819 1/20 0.41
CSF1R P07333 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3511705 0.81 PARP1 (0.47) ALDH1A1KDM4EHPGDMAPTTSHR
SCHEMBL8578585 0.77 ALDH1A1 (0.57) ALDH1A1KDM4EHPGDMAPTTSHR
SCHEMBL8580566 0.76 ERN1 (0.40) ALDH1A1KDM4EHPGDMAPTTSHR
SCHEMBL29951147 0.76 KDM4E (0.57) ALDH1A1KDM4EHPGDMAPTTSHR
SCHEMBL28257533 0.76 ALDH1A1 (0.44) ALDH1A1KDM4EHPGDMAPTTSHR
SCHEMBL15210226 0.76 ERN1 (0.44) ALDH1A1KDM4EHPGDMAPTTSHR
SCHEMBL4967588 0.75 ALDH1A1 (0.70) ALDH1A1KDM4EHPGDMAPTTSHR
SCHEMBL27700719 0.75 ALDH1A1 (0.70) ALDH1A1KDM4EHPGDMAPTTSHR
SCHEMBL39118 0.75 ALDH1A1 (0.70) ALDH1A1KDM4EHPGDMAPTTSHR
SCHEMBL8582279 0.75 THRB (0.41) ALDH1A1KDM4EHPGDMAPTTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5792840-A SUBSTITUTED GLUCOPYRANOSYL PHOSPHATES SANKYO COMPANY, LIMITED (JP) 1998-08-11 US disclosed
EP-0437016-B1 Lipid A analogues having immunoactivating and anti-tumour activity SANKYO CO (JP) 1996-05-01 EP disclosed
EP-0437016-A2 Lipid A analogues having immunoactivating and anti-tumour activity Sankyo Company Limited (JP) 1991-07-17 EP disclosed