SCHEMBL8580642

SCHEMBL8580642

CC(C)(C)c1cc(C=C2NC(=O)CS2)cc(C(C)(C)C)c1O

nearest known ligand 0.57

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 10/20 0.57
PTGS1 P23219 7/20 0.57
CYP1A2 P05177 1/20 0.56
CYP2C9 P11712 1/20 0.56
GAA P10253 2/20 0.52
ALOX5 P09917 2/20 0.50
EEF2K O00418 1/20 0.50
SRC P12931 1/20 0.50
MEN1 O00255 1/20 0.47
ALDH1A1 P00352 1/20 0.47
KMT2A Q03164 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8581179 0.92 PTGS2 (0.49) PTGS2PTGS1CYP1A2CYP2C9GAA
SCHEMBL8580941 0.85 TP53 (0.45) PTGS2PTGS1CYP1A2CYP2C9ALDH1A1
SCHEMBL8580718 0.80 MAPT (0.42) PTGS2PTGS1CYP1A2CYP2C9GAA
SCHEMBL8582453 0.77 CYP1A2 (0.56) PTGS2PTGS1CYP1A2ALDH1A1
Darbufelone SCHEMBL452950 0.73 PTGS2 (0.75) PTGS2PTGS1CYP1A2CYP2C9GAA
Darbufelone SCHEMBL8526046 0.73 PTGS2 (0.75) PTGS2PTGS1CYP1A2CYP2C9GAA
Darbufelone SCHEMBL452951 0.73 PTGS2 (0.75) PTGS2PTGS1CYP1A2CYP2C9GAA
SCHEMBL3667218 0.72 PTGS2 (1.00) PTGS2PTGS1GAAALOX5
SCHEMBL3667216 0.72 PTGS2 (1.00) PTGS2PTGS1GAAALOX5
SCHEMBL8962138 0.72 PTGS2 (1.00) PTGS2PTGS1GAAALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5731336-A USING ARYL-SUBSTITUTED RHODAMINES ELI LILLY AND COMPANY (US) 1998-03-24 US disclosed