SCHEMBL8580718

SCHEMBL8580718

CC(C)(C)c1cc(CC=C2NC(=O)CS2)cc(C(C)(C)C)c1O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.42
MAPK1 P28482 3/20 0.42
TP53 P04637 2/20 0.42
NFKB1 P19838 2/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
NFKB2 Q00653 1/20 0.42
RELA Q04206 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
ALDH1A1 P00352 5/20 0.41
CYP1A2 P05177 3/20 0.41
KMT2A Q03164 3/20 0.41
TSHR P16473 3/20 0.41
MEN1 O00255 2/20 0.41
CYP3A4 P08684 2/20 0.41
BLM P54132 2/20 0.41
ATM Q13315 2/20 0.41
HIF1A Q16665 2/20 0.41
NPSR1 Q6W5P4 2/20 0.41
USP2 O75604 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8580642 0.80 PTGS2 (0.57) ALDH1A1CYP1A2KMT2AMEN1PTGS2
SCHEMBL8991939 0.74 PTGS2 (0.44) MAPTMAPK1TP53NFKB1ALDH1A1
SCHEMBL9027935 0.74 PTGS2 (0.44) MAPTMAPK1TP53NFKB1ALDH1A1
SCHEMBL8580713 0.73 ALDH1A1 (0.42) MAPTMAPK1TP53NFKB1ALDH1A1
SCHEMBL8581179 0.73 PTGS2 (0.49) MAPTMAPK1TP53NFKB1NPC1
SCHEMBL8580941 0.71 TP53 (0.45) MAPTMAPK1TP53NFKB1NPC1
SCHEMBL8895700 0.70 ALDH1A1 (0.42) MAPTMAPK1TP53NFKB1ALDH1A1
SCHEMBL8580683 0.70 ALDH1A1 (0.40) MAPTMAPK1SMN1; SMN2ALDH1A1CYP1A2
SCHEMBL4729051 0.69 ALDH1A1 (0.65) MAPTMAPK1TP53NFKB1SMN1; SMN2
SCHEMBL8908613 0.69 PTGS2 (0.41) MAPTMAPK1TP53NFKB1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5731336-A USING ARYL-SUBSTITUTED RHODAMINES ELI LILLY AND COMPANY (US) 1998-03-24 US disclosed