SCHEMBL8580669

SCHEMBL8580669

CC(C)(C)C(=O)C[C@@H](NC(=O)C(C)(C)C)C(O)=S

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.32
CNR2 P34972 1/20 0.31
POLB P06746 1/20 0.31
MAPK1 P28482 1/20 0.31
RECQL P46063 1/20 0.31
CYP2C9 P11712 3/20 0.30
CYP2C19 P33261 3/20 0.30
ALDH1A1 P00352 2/20 0.30
CYP1A2 P05177 2/20 0.30
CYP3A4 P08684 2/20 0.30
KDM4E B2RXH2 1/20 0.30
GAA P10253 1/20 0.30
HPGD P15428 1/20 0.30
TAAR1 Q96RJ0 1/20 0.30
NPC1 O15118 1/20 0.30
ALOX12 P18054 1/20 0.30
RAB9A P51151 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
CYP2D6 P10635 1/20 0.30
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8582124 0.85 SMN1; SMN2 (0.41) SMN1; SMN2RECQLALDH1A1KDM4E
SCHEMBL25928849 0.85 ACE (0.36) SMN1; SMN2CNR2POLBMAPK1RECQL
SCHEMBL8580667 0.79 CNR2 (0.32) CNR2NPSR1
SCHEMBL25928846 0.78 NPSR1 (0.37) SMN1; SMN2CNR2NPSR1
SCHEMBL24263122 0.72 CNR2 (0.34) CNR2POLBMAPK1CYP2C9CYP2C19
SCHEMBL24263116 0.72 CNR2 (0.34) CNR2POLBMAPK1CYP2C9CYP2C19
SCHEMBL19756282 0.71 GRIA1 (0.44)
SCHEMBL20623017 0.71 GRIA1 (0.37) TSHR
SCHEMBL24263148 0.71 CNR2 (0.37) CNR2POLBMAPK1NPSR1
SCHEMBL15605968 0.71 CA2 (0.47) GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5705527-A VASODILATORS AND ANGINA PECTORIS SANKYO COMPANY, LIMITED (JP) 1998-01-06 US disclosed
EP-0641769-B1 AMINO ACID DERIVATIVE SANKYO CO (JP) 1997-01-29 EP disclosed
EP-0641769-A1 AMINO ACID DERIVATIVE SANKYO COMPANY LIMITED (JP) 1995-03-08 EP disclosed