SCHEMBL8580793

SCHEMBL8580793

CS(=O)(=O)N1c2ccc(F)cc2C2(CCNCC2)[C@@H]1C(=O)OCc1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GNRHR P30968 2/20 0.41
KCNH2 Q12809 1/20 0.41
CASP1 P29466 1/20 0.37
PKM P14618 1/20 0.36
ELANE P08246 3/20 0.35
F2 P00734 1/20 0.35
CTSG P08311 1/20 0.35
HTR2C P28335 1/20 0.35
MGAT2 Q10469 1/20 0.34
TACR1 P25103 1/20 0.34
GRM5 P41594 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8707482 0.89 HTR2C (0.38) ELANEF2CTSGHTR2CTACR1
SCHEMBL7542146 0.70 NPC1 (0.43) CASP1HTR2CMGAT2TACR1GRM5
SCHEMBL16539832 0.67 HTR2C (0.43) HTR2C
SCHEMBL8067334 0.67 TACR1 (0.57) TACR1
SCHEMBL29661999 0.67 TACR1 (0.57) TACR1
SCHEMBL5783726 0.65 GNRHR (0.43) GNRHRKCNH2HTR2C
SCHEMBL1670310 0.64 HTR2C (0.49) HTR2CTACR1
SCHEMBL5600502 0.64 GNRHR (0.47) GNRHRKCNH2HTR2C
Alcohol SCHEMBL27541427 0.64 TSHR (0.53) PKMHTR2C
Hydrochloric Acid SCHEMBL8814693 0.64 BACE1 (0.45) HTR2CTACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998025605-A1 SPIRO-SUBSTITUTED AZACYCLES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY MERCK & CO., INC. (US) 1998-06-18 WO claimed