SCHEMBL8707482

SCHEMBL8707482

CS(=O)(=O)N1c2ccccc2C2(CCNCC2)C1C(=O)OCc1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 1/20 0.38
ELANE P08246 7/20 0.37
TACR1 P25103 1/20 0.37
BACE1 P56817 1/20 0.37
TSHR P16473 1/20 0.36
F2 P00734 1/20 0.36
CTSG P08311 1/20 0.36
NPC1 O15118 1/20 0.36
GAA P10253 1/20 0.36
MAPK1 P28482 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8580793 0.89 GNRHR (0.41) HTR2CELANETACR1F2CTSG
SCHEMBL16539832 0.78 HTR2C (0.43) HTR2CNPC1GAAMAPK1RAB9A
SCHEMBL8469385 0.76 GHSR (0.56) TACR1
SCHEMBL7500323 0.76 GHSR (0.55) TACR1
SCHEMBL1670310 0.74 HTR2C (0.49) HTR2CTACR1NPC1GAAMAPK1
SCHEMBL8328802 0.74 GNRHR (0.40) HTR2CGAA
SCHEMBL6649033 0.73 HTR2C (0.40) HTR2CELANENPC1GAAMAPK1
Hydrochloric Acid SCHEMBL8814693 0.70 BACE1 (0.45) HTR2CTACR1BACE1TSHRNPC1
SCHEMBL5598985 0.67 MTNR1A (0.36) HTR2CMAPK1
SCHEMBL24433396 0.67 TSHR (0.43) HTR2CTACR1BACE1TSHRGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998018762-A1 NEW DERIVATIVES OF DIVERSELY SUBSTITUTED CYCLICAL AMIDE SELECTIVE ANTAGONISTS OF THE HUMAN RECEPTOR NK3, PROCESS FOR OBTAINING THEM, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SANOFI (FR) 1998-05-07 WO disclosed