SCHEMBL8580902

SCHEMBL8580902

COC(=O)Cc1c(-c2ccc3c(c2)OCO3)c2ccccc2n(Cc2ccccc2OC)c1=O

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EDNRB P24530 11/20 0.75
EDNRA P25101 4/20 0.49
ALDH1A1 P00352 3/20 0.47
MAPK1 P28482 2/20 0.47
HPGD P15428 1/20 0.47
MAPT P10636 1/20 0.44
RXFP1 Q9HBX9 1/20 0.44
LMNA P02545 2/20 0.44
CYP1A2 P05177 2/20 0.44
CYP3A4 P08684 2/20 0.44
CYP2D6 P10635 2/20 0.44
CYP2C9 P11712 2/20 0.44
CYP2C19 P33261 2/20 0.44
HSD17B10 Q99714 2/20 0.44
CLK4 Q9HAZ1 2/20 0.44
ALOX15 P16050 1/20 0.44
TSHR P16473 1/20 0.44
HIF1A Q16665 1/20 0.44
MEN1 O00255 1/20 0.44
USP2 O75604 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6314927 0.92 EDNRB (0.79) EDNRBEDNRAALDH1A1MAPK1HPGD
SCHEMBL6315635 0.86 EDNRB (1.00) EDNRBEDNRAALDH1A1
SCHEMBL8798255 0.83 EDNRB (0.79) EDNRBEDNRAALDH1A1MAPK1HPGD
SCHEMBL6314851 0.77 EDNRB (0.75) EDNRBEDNRAMAPTTSHRMEN1
SCHEMBL8578004 0.77 EDNRB (0.86) EDNRBEDNRA
SCHEMBL8577096 0.76 EDNRB (0.85) EDNRBEDNRAALDH1A1MAPK1HPGD
SCHEMBL795880 0.76 EDNRB (1.00) EDNRBEDNRA
SCHEMBL8797682 0.75 EDNRB (0.78) EDNRBEDNRAMAPT
SCHEMBL8576085 0.75 EDNRB (1.00) EDNRBEDNRA
SCHEMBL8799108 0.75 EDNRB (0.77) EDNRBEDNRAALDH1A1MAPK1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5731321-A Endothelin receptor antagonists MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1998-03-24 US disclosed