SCHEMBL8799108

SCHEMBL8799108

COC(=O)Oc1c(-c2ccc3c(c2)OCO3)c2c(OC)c(OC)ccc2n(Cc2ccccc2OC)c1=O

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EDNRB P24530 12/20 0.77
EDNRA P25101 4/20 0.44
ALDH1A1 P00352 3/20 0.44
MAPK1 P28482 2/20 0.44
HPGD P15428 2/20 0.44
KDM4E B2RXH2 2/20 0.42
MAPT P10636 2/20 0.42
NPSR1 Q6W5P4 1/20 0.42
CYP3A4 P08684 3/20 0.40
HSD17B10 Q99714 3/20 0.40
USP2 O75604 2/20 0.40
CYP1A2 P05177 2/20 0.40
CYP2D6 P10635 2/20 0.40
ALOX15 P16050 2/20 0.40
TSHR P16473 2/20 0.40
CYP2C19 P33261 2/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
MCHR1 Q99705 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8799772 0.94 EDNRB (0.68) EDNRBEDNRAALDH1A1HPGDKDM4E
SCHEMBL8798950 0.92 EDNRB (0.81) EDNRBEDNRAALDH1A1MAPK1HPGD
SCHEMBL8798090 0.91 EDNRB (0.64) EDNRBEDNRAALDH1A1HPGDKDM4E
SCHEMBL8799661 0.89 EDNRB (0.61) EDNRBEDNRAALDH1A1MAPK1KDM4E
SCHEMBL8577096 0.88 EDNRB (0.85) EDNRBEDNRAALDH1A1MAPK1HPGD
SCHEMBL8576085 0.87 EDNRB (1.00) EDNRBEDNRA
SCHEMBL8798300 0.86 EDNRB (0.71) EDNRBEDNRAALDH1A1KDM4EMAPT
SCHEMBL8798655 0.83 EDNRB (0.67) EDNRBEDNRAALDH1A1HPGDKDM4E
SCHEMBL8797682 0.83 EDNRB (0.78) EDNRBEDNRAMAPTTP53
SCHEMBL8578545 0.82 EDNRB (0.75) EDNRBEDNRAALDH1A1MAPK1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0757039-A1 Endothelin receptor antagonists MERCK PATENT GmbH (DE) 1997-02-05 EP disclosed