SCHEMBL8583129

SCHEMBL8583129

COC(=O)c1ccc(C2CCCC2)c(S(C)(=O)=O)c1Br

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
YAP1 P46937 1/20 0.37
KDM4E B2RXH2 8/20 0.36
ALDH1A1 P00352 5/20 0.36
HSD17B10 Q99714 3/20 0.36
HPGD P15428 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
PDK2 Q15119 1/20 0.35
PDK4 Q16654 1/20 0.35
PTGS2 P35354 1/20 0.34
TSHR P16473 1/20 0.34
RECQL P46063 1/20 0.34
KMT2A Q03164 2/20 0.33
RIPK1 Q13546 1/20 0.33
RBP4 P02753 1/20 0.33
OPRK1 P41145 1/20 0.33
MEN1 O00255 1/20 0.33
MAPK1 P28482 1/20 0.33
PTGDR Q13258 1/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8578768 0.99 YAP1 (0.39) YAP1KDM4EALDH1A1HSD17B10HPGD
SCHEMBL8583575 0.95 PDK2 (0.39) YAP1KDM4EALDH1A1HSD17B10HPGD
SCHEMBL8585348 0.90 ALDH1A1 (0.38) KDM4EALDH1A1HSD17B10HPGDSMN1; SMN2
SCHEMBL8580491 0.85 CMA1 (0.40) YAP1KDM4EALDH1A1HSD17B10HPGD
SCHEMBL8581200 0.84 ALOX5AP (0.37) YAP1KDM4EALDH1A1HSD17B10HPGD
SCHEMBL8579027 0.84 YAP1 (0.39) YAP1KDM4EALDH1A1HSD17B10HPGD
SCHEMBL8581857 0.84 YAP1 (0.37) YAP1KDM4EALDH1A1HSD17B10HPGD
SCHEMBL8582273 0.83 YAP1 (0.39) YAP1KDM4EALDH1A1HSD17B10HPGD
SCHEMBL8580134 0.83 YAP1 (0.39) YAP1KDM4EALDH1A1HSD17B10HPGD
SCHEMBL8583191 0.83 KDM4E (0.36) YAP1KDM4EALDH1A1HSD17B10HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5840761-A Alkylbenzoylguanidine derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1998-11-24 US disclosed