SCHEMBL8583772

SCHEMBL8583772

O=C(O)Nc1cccc2cccnc12.O=S(=O)(Nc1cccc2cccnc12)c1ccc2ccccc2c1

nearest known ligand 0.82

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 8/20 0.82
GLO1 Q04760 7/20 0.82
KMT2A Q03164 6/20 0.82
MEN1 O00255 5/20 0.82
SLC40A1 Q9NP59 9/20 0.65
AGTR1 P30556 2/20 0.65
G6PD P11413 1/20 0.65
NFKBIA P25963 1/20 0.65
METAP2 P50579 1/20 0.65
METAP1 P53582 1/20 0.65
PAX8 Q06710 1/20 0.65
ATM Q13315 1/20 0.65
MITF O75030 1/20 0.61
S1PR4 O95977 1/20 0.61
ALDH1A1 P00352 1/20 0.61
LMNA P02545 1/20 0.61
MAPT P10636 1/20 0.61
S1PR1 P21453 1/20 0.61
OPRK1 P41145 1/20 0.61
HTT P42858 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6979087 0.91 TDP1 (1.00) TDP1GLO1KMT2AMEN1SLC40A1
SCHEMBL442367 0.80 SLC40A1 (1.00) TDP1GLO1KMT2AMEN1SLC40A1
SCHEMBL1695444 0.80 KDR (0.71) TDP1KMT2AMEN1ALDH1A1MAPT
SCHEMBL29851236 0.80 KDR (0.71) TDP1KMT2AMEN1ALDH1A1MAPT
SCHEMBL23413185 0.80 MEN1 (0.67) TDP1GLO1KMT2AMEN1SLC40A1
SCHEMBL30092884 0.80 MEN1 (0.67) TDP1GLO1KMT2AMEN1SLC40A1
SCHEMBL7746129 0.79 SLC40A1 (0.97) TDP1GLO1KMT2AMEN1SLC40A1
SCHEMBL30925435 0.78 SLC40A1 (0.74) TDP1GLO1KMT2AMEN1SLC40A1
SCHEMBL16750883 0.78 SLC40A1 (0.74) TDP1GLO1KMT2AMEN1SLC40A1
SCHEMBL12964661 0.78 SLC40A1 (0.75) TDP1GLO1KMT2AMEN1SLC40A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999029670-A2 AMINOCARBONYLTETRALIN AND DIHYDRONAPHTALENE DERIVATES AS THROMBIN INHIBITORS BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-06-17 WO disclosed