SCHEMBL8585368

SCHEMBL8585368

CNCCC[C@@H](C(=O)NC(=N)N)N(Cc1ccc(O)cc1)C(=O)C(c1ccccc1)c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NPY1R P25929 13/20 0.40
CNR1 P21554 1/20 0.37
CNR2 P34972 1/20 0.37
NPFFR1 Q9GZQ6 2/20 0.36
NPFFR2 Q9Y5X5 2/20 0.36
NPY5R Q15761 2/20 0.36
TDP1 Q9NUW8 1/20 0.36
HTR2A P28223 1/20 0.36
HRH1 P35367 1/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
NPY4R P50391 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7043232 0.88 TDP1 (0.40) NPY1RCNR1CNR2NPFFR1NPFFR2
SCHEMBL8127029 0.83 NPY1R (0.41) NPY1RCNR1CNR2NPFFR1NPFFR2
SCHEMBL9195693 0.82 NPY1R (0.42) NPY1RCNR1CNR2NPFFR1NPFFR2
SCHEMBL1593414 0.82 NPY1R (0.42) NPY1RCNR1CNR2NPFFR1NPFFR2
SCHEMBL4650863 0.80 NPY1R (0.40) NPY1RCNR1CNR2NPFFR1NPFFR2
SCHEMBL7753050 0.80 NPY1R (0.43) NPY1RCNR1CNR2NPFFR1NPFFR2
SCHEMBL8126197 0.80 NPY1R (0.43) NPY1RCNR1CNR2NPFFR1NPFFR2
SCHEMBL8119315 0.78 NPY1R (0.42) NPY1RCNR1CNR2NPFFR1NPFFR2
SCHEMBL8527836 0.78 NPY1R (0.43) NPY1RNPFFR1NPFFR2NPY5RTDP1
SCHEMBL8112714 0.77 MEN1 (0.42) CNR1CNR2TDP1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0885186-A1 AMINO ACID DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS AND PROCESSES FOR PREPARING THEM Dr. Karl Thomae GmbH (DE) 1998-12-23 EP disclosed
WO-1997019911-A1 AMINO ACID DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS AND PROCESSES FOR PREPARING THEM DR. KARL THOMAE GMBH (DE) 1997-06-05 WO disclosed