Terofenamate

Terofenamate

SCHEMBL8585656

CCOCOC(=O)c1ccccc1Nc1c(Cl)ccc(C)c1Cl.O=C(O)c1ccccc1Nc1cccc(C(F)(F)F)c1

nearest known ligand 0.59

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Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
METTL3 Q86U44 2/20 0.59
PTGS2 P35354 4/20 0.54
AKR1C3 P42330 2/20 0.54
AKR1C2 P52895 2/20 0.54
TTR P02766 2/20 0.54
MEN1 O00255 1/20 0.54
AKR1B10 O60218 1/20 0.54
ABCB11 O95342 1/20 0.54
ADORA3 P0DMS8 1/20 0.54
CHRM1 P11229 1/20 0.54
FABP2 P12104 1/20 0.54
RXRA P19793 1/20 0.54
TBXA2R P21731 1/20 0.54
NR4A1 P22736 1/20 0.54
PTGS1 P23219 1/20 0.54
PDE4A P27815 1/20 0.54
MAPK1 P28482 1/20 0.54
NR4A2 P43354 1/20 0.54
KMT2A Q03164 1/20 0.54
AKR1C1 Q04828 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Flufenamic Acid SCHEMBL21408198 0.88 PTGS2 (0.69) METTL3PTGS2AKR1C3AKR1C2TTR
Terofenamate SCHEMBL49245 0.84 METTL3 (0.83) METTL3PTGS2AKR1C3AKR1C2TTR
Terofenamate SCHEMBL9856559 0.84 METTL3 (0.81) METTL3PTGS2AKR1C3AKR1C2TTR
Terofenamate SCHEMBL26088 0.84 METTL3 (0.84) METTL3PTGS2AKR1C3AKR1C2TTR
Terofenamate SCHEMBL29483481 0.84 METTL3 (0.84) METTL3PTGS2AKR1C3AKR1C2TTR
Terofenamate SCHEMBL20503838 0.83 METTL3 (0.70) METTL3PTGS2AKR1C3AKR1C2TTR
Terofenamate SCHEMBL9445147 0.83 METTL3 (0.70) METTL3PTGS2AKR1C3AKR1C2TTR
Terofenamate SCHEMBL7160746 0.83 METTL3 (0.79) METTL3PTGS2AKR1C3AKR1C2TTR
Terofenamate SCHEMBL16760954 0.83 METTL3 (0.79) METTL3PTGS2AKR1C3AKR1C2TTR
Terofenamate SCHEMBL1671593 0.83 METTL3 (0.83) METTL3PTGS2AKR1C3AKR1C2TTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0759750-A4 COMPOSITIONS FOR TREATMENT OF CHRONIC INFLAMMATORY DISEASES SHAPIRO HOWARD K (US) 1998-05-27 EP claimed
EP-0759750-A1 COMPOSITIONS FOR TREATMENT OF CHRONIC INFLAMMATORY DISEASES SHAPIRO, Howard, K. (US) 1997-03-05 EP claimed
WO-1995031194-A1 COMPOSITIONS FOR TREATMENT OF CHRONIC INFLAMMATORY DISEASES SHAPIRO HOWARD K (US) 1995-11-23 WO claimed