SCHEMBL8585682

SCHEMBL8585682

Oc1cccnc1-n1ccnc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.58
CYP3A4 P08684 5/20 0.49
TDP1 Q9NUW8 4/20 0.49
CYP1A2 P05177 3/20 0.49
TSHR P16473 2/20 0.49
ENPP2 Q13822 1/20 0.47
MKNK1 Q9BUB5 1/20 0.47
MKNK2 Q9HBH9 1/20 0.47
CYP2A6 P11509 1/20 0.46
NCOA3 Q9Y6Q9 1/20 0.45
LMNA P02545 4/20 0.41
MAPT P10636 2/20 0.41
KDM4E B2RXH2 1/20 0.41
BRD4 O60885 1/20 0.41
POLB P06746 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
ALOX15 P16050 1/20 0.41
ELANE P08246 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20394478 0.81 CYP3A4 (0.46) IDO1CYP3A4TDP1CYP1A2TSHR
SCHEMBL2592326 0.80 L3MBTL1 (0.42) IDO1TSHRLMNAMAPTKDM4E
SCHEMBL22556880 0.78 LMNA (0.47) IDO1CYP3A4TDP1CYP1A2TSHR
SCHEMBL22719451 0.76 MYC (0.54) CYP3A4TDP1CYP1A2TSHRCYP2A6
SCHEMBL6306259 0.75 CYP3A4 (0.43) IDO1CYP3A4TDP1CYP1A2TSHR
SCHEMBL15881144 0.75 CYP3A4 (0.53) IDO1CYP3A4TDP1CYP1A2TSHR
SCHEMBL10761274 0.74 CYP3A4 (0.50) CYP3A4TDP1CYP1A2TSHRMKNK1
SCHEMBL3273101 0.74 NCOA3 (0.45) IDO1CYP3A4TDP1CYP1A2TSHR
SCHEMBL29523312 0.73 IDO1 (1.00) IDO1CYP3A4TDP1CYP1A2TSHR
SCHEMBL57158 0.73 IDO1 (1.00) IDO1CYP3A4TDP1CYP1A2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0857171-A2 IMIDAZOLE DERIVATIVES AND THE USE THEREOF AS NITROGEN MONOXIDE SYNTHASE INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 1998-08-12 EP disclosed
WO-1997015555-A2 IMIDAZOLE DERIVATIVES AND THE USE THEREOF AS NITROGEN MONOXIDE SYNTHASE INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 1997-05-01 WO disclosed