SCHEMBL8585740

SCHEMBL8585740

CC(N)C(=O)Nc1cccnc1OOC(=O)C1(NC(=O)OC(C)(C)C)CCc2ccccc2C1

nearest known ligand 0.45

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GHSR Q92847 2/20 0.45
P2RY1 P47900 9/20 0.35
BACE1 P56817 2/20 0.34
CYP3A4 P08684 3/20 0.32
SCN9A Q15858 3/20 0.32
PYGL P06737 1/20 0.32
SCN10A Q9Y5Y9 2/20 0.32
XIAP P98170 2/20 0.32
METAP1 P53582 1/20 0.31
BIRC2 Q13490 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8581721 0.88 GHSR (0.48) GHSRBACE1PYGLXIAP
SCHEMBL8613091 0.84 GHSR (0.40) GHSRCYP3A4SCN9A
SCHEMBL8580708 0.74 GHSR (0.43) GHSRBACE1
SCHEMBL5196233 0.73 GHSR (0.61) GHSRBACE1PYGL
SCHEMBL8583068 0.72 GHSR (0.43) GHSR
SCHEMBL2813574 0.71 GHSR (0.63) GHSRBACE1PYGL
SCHEMBL18614234 0.71 GHSR (0.63) GHSRBACE1PYGL
SCHEMBL29715495 0.71 GHSR (0.63) GHSRBACE1PYGL
SCHEMBL8997810 0.70 P2RY1 (0.39) P2RY1
SCHEMBL8584168 0.70 BUB1 (0.32) GHSRP2RY1BACE1CYP3A4SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5837807-A DIPEPTIDES AND CYCLIC PEPTIDE DERIVATIVES OF AMINO TETRAHYDRONAPHTHALENECARBOXYLIC ACID AND HELICAL DOMAINS HOFFMANN-LA ROCHE INC. (US) 1998-11-17 US disclosed