SCHEMBL8613091

SCHEMBL8613091

CC(NC(=O)OCc1ccccc1)C(=O)NC(C)C(=O)Nc1cccnc1OOC(=O)[C@]1(NC(=O)OC(C)(C)C)CCc2ccccc2C1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GHSR Q92847 2/20 0.40
SYK P43405 1/20 0.39
JAK2 O60674 1/20 0.37
CTSK P43235 1/20 0.36
PSMB5 P28074 1/20 0.36
HDAC1 Q13547 5/20 0.35
HDAC4 P56524 3/20 0.35
HDAC6 Q9UBN7 3/20 0.35
NTSR1 P30989 1/20 0.35
MAPT P10636 1/20 0.35
MAPK1 P28482 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
CYP3A4 P08684 1/20 0.35
SCN9A Q15858 1/20 0.35
POLB P06746 1/20 0.34
ELANE P08246 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8583068 0.90 GHSR (0.43) GHSRSYKJAK2CTSKPSMB5
SCHEMBL8585740 0.84 GHSR (0.45) GHSRCYP3A4SCN9A
SCHEMBL8582291 0.81 SYK (0.42) GHSRSYKCTSKPSMB5NTSR1
SCHEMBL8997804 0.79 P2RY1 (0.37) SYKJAK2CTSKHDAC1HDAC4
SCHEMBL8581721 0.72 GHSR (0.48) GHSRMAPTL3MBTL1POLB
SCHEMBL8997594 0.71 SYK (0.40) SYKJAK2CTSKPSMB5MAPT
SCHEMBL8582293 0.70 SYK (0.44) GHSRSYKCTSKPSMB5NTSR1
SCHEMBL8845144 0.70 GHSR (0.39) GHSRSYKL3MBTL1POLB
SCHEMBL8580708 0.69 GHSR (0.43) GHSR
SCHEMBL8997810 0.69 P2RY1 (0.39) MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5837807-A DIPEPTIDES AND CYCLIC PEPTIDE DERIVATIVES OF AMINO TETRAHYDRONAPHTHALENECARBOXYLIC ACID AND HELICAL DOMAINS HOFFMANN-LA ROCHE INC. (US) 1998-11-17 US disclosed